| Reaction Details |
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 | Report a problem with these data |
| Target | Lysophosphatidic acid receptor 1 |
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| Ligand | BDBM50539029 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1977566 (CHEMBL4610701) |
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| EC50 | 3600±n/a nM |
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| Citation |  González-Gil, I; Zian, D; Vázquez-Villa, H; Hernández-Torres, G; Martínez, RF; Khiar-Fernández, N; Rivera, R; Kihara, Y; Devesa, I; Mathivanan, S; Del Valle, CR; Zambrana-Infantes, E; Puigdomenech, M; Cincilla, G; Sanchez-Martinez, M; Rodríguez de Fonseca, F; Ferrer-Montiel, AV; Chun, J; López-Vales, R; López-Rodríguez, ML; Ortega-Gutiérrez, S A Novel Agonist of the Type 1 Lysophosphatidic Acid Receptor (LPA J Med Chem63:2372-2390 (2020) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Lysophosphatidic acid receptor 1 |
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| Name: | Lysophosphatidic acid receptor 1 |
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| Synonyms: | EDG2 | LPA receptor 1 | LPA-1 | LPA1 | LPAR1 | LPAR1_HUMAN | Lysophosphatidic acid receptor 1 (LPA1) | Lysophosphatidic acid receptor Edg-2 |
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| Type: | Enzyme |
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| Mol. Mass.: | 41120.55 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Q92633 |
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| Residue: | 364 |
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| Sequence: | MAAISTSIPVISQPQFTAMNEPQCFYNESIAFFYNRSGKHLATEWNTVSKLVMGLGITVC
IFIMLANLLVMVAIYVNRRFHFPIYYLMANLAAADFFAGLAYFYLMFNTGPNTRRLTVST
WLLRQGLIDTSLTASVANLLAIAIERHITVFRMQLHTRMSNRRVVVVIVVIWTMAIVMGA
IPSVGWNCICDIENCSNMAPLYSDSYLVFWAIFNLVTFVVMVVLYAHIFGYVRQRTMRMS
RHSSGPRRNRDTMMSLLKTVVIVLGAFIICWTPGLVLLLLDVCCPQCDVLAYEKFFLLLA
EFNSAMNPIIYSYRDKEMSATFRQILCCQRSENPTGPTEGSDRSASSLNHTILAGVHSND
HSVV
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| BDBM50539029 |
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| n/a |
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| Name | BDBM50539029 |
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| Synonyms: | CHEMBL4646443 |
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| Type | Small organic molecule |
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| Emp. Form. | C17H22N2 |
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| Mol. Mass. | 254.37 |
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| SMILES | CC1CCC2(C)N(CCc3c2[nH]c2ccccc32)C1 |
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| Structure | 
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