| Reaction Details |
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 | Report a problem with these data |
| Target | Casein kinase 1, delta tv1 |
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| Ligand | BDBM50364141 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1985499 (CHEMBL4618905) |
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| IC50 | 7.7±n/a nM |
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| Citation |  Cescon, E; Bolcato, G; Federico, S; Bissaro, M; Valentini, A; Ferlin, MG; Spalluto, G; Sturlese, M; Moro, S Scaffold Repurposing of in-House Chemical Library toward the Identification of New Casein Kinase 1 ? Inhibitors. ACS Med Chem Lett11:1168-1174 (2020) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Casein kinase 1, delta tv1 |
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| Name: | Casein kinase 1, delta tv1 |
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| Synonyms: | CSNK1D |
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| Type: | PROTEIN |
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| Mol. Mass.: | 47258.61 |
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| Organism: | Sus scrofa |
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| Description: | ChEMBL_106594 |
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| Residue: | 415 |
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| Sequence: | MELRVGNRYRLGRKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQ
GGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIH
SKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYA
SINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVL
CKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNMLKFGASRA
ADDAERERRDREERLRHSRNPATRGLPSTASGRLRGTQEAAPPTPLTPTSHTANTSPRPV
SGMERERKVSMRLHRGAPVNISSSDLTGRQDTSRMSTSQIAGRVAASGLQSAVHR
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| BDBM50364141 |
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| n/a |
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| Name | BDBM50364141 |
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| Synonyms: | CHEMBL1951415 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H20FN5 |
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| Mol. Mass. | 337.394 |
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| SMILES | Nc1nccc(n1)-c1c(ncn1C1CCCCC1)-c1ccc(F)cc1 |
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| Structure | 
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