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TargetLeukotriene B4 receptor 2
LigandBDBM50212626
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1993331 (CHEMBL4627066)
IC50 150±n/a nM
Citation Kim, MWei, JDHarmalkar, DSGoo, JILee, KChoi, YKim, JHCho, AE Elucidation of Mechanism for Ligand Efficacy at Leukotriene B ACS Med Chem Lett11:1529-1534 (2020) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Leukotriene B4 receptor 2
Name:Leukotriene B4 receptor 2
Synonyms:BLT2R | BLTR2 | LT4R2_HUMAN | LTB4 receptor JULF2 | LTB4-R 2 | LTB4-R2 | LTB4R2 | LTB4R2 protein | Leukotriene B4 | Leukotriene B4 R2 | Leukotriene B4 receptor | Leukotriene B4 receptor 2 | Leukotriene B4 receptor BLT2 | Leukotriene b1 | Seven transmembrane receptor BLTR2
Type:Enzyme Catalytic Domain
Mol. Mass.:37964.86
Organism:Homo sapiens (Human)
Description:Leukotriene 2 0 HUMAN::Q9NPC1
Residue:358
Sequence:
MSVCYRPPGNETLLSWKTSRATGTAFLLLAALLGLPGNGFVVWSLAGWRPARGRPLAATL
VLHLALADGAVLLLTPLFVAFLTRQAWPLGQAGCKAVYYVCALSMYASVLLTGLLSLQRC
LAVTRPFLAPRLRSPALARRLLLAVWLAALLLAVPAAVYRHLWRDRVCQLCHPSPVHAAA
HLSLETLTAFVLPFGLMLGCYSVTLARLRGARWGSGRHGARVGRLVSAIVLAFGLLWAPY
HAVNLLQAVAALAPPEGALAKLGGAGQAARAGTTALAFFSSSVNPVLYVFTAGDLLPRAG
PRFLTRLFEGSGEARGGGRSREGTMELRTTPQLKVVGQGRGNGDPGGGMEKDGPEWDL
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50212626
n/a
NameBDBM50212626
Synonyms:LY-255283
TypeSmall organic molecule
Emp. Form.C19H28N4O3
Mol. Mass.360.4506
SMILESCCc1cc(C(C)=O)c(O)cc1OCCCCCC(C)(C)c1nn[nH]n1
Structure
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