| Reaction Details |
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 | Report a problem with these data |
| Target | P2Y purinoceptor 1 |
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| Ligand | BDBM50102301 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_147891 (CHEMBL884926) |
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| IC50 | 100000±n/a nM |
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| Citation |  Kim, YC; Brown, SG; Harden, TK; Boyer, JL; Dubyak, G; King, BF; Burnstock, G; Jacobson, KA Structure-activity relationships of pyridoxal phosphate derivatives as potent and selective antagonists of P2X1 receptors. J Med Chem44:340-9 (2001) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| P2Y purinoceptor 1 |
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| Name: | P2Y purinoceptor 1 |
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| Synonyms: | P2RY1 | P2RY1_MELGA |
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| Type: | n/a |
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| Mol. Mass.: | 41199.64 |
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| Organism: | Meleagris gallopavo |
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| Description: | n/a |
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| Residue: | 362 |
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| Sequence: | MTEALISAALNGTQPELLAGGWAAGNASTKCSLTKTGFQFYYLPTVYILVFITGFLGNSV
AIWMFVFHMRPWSGISVYMFNLALADFLYVLTLPALIFYYFNKTDWIFGDVMCKLQRFIF
HVNLYGSILFLTCISVHRYTGVVHPLKSLGRLKKKNAVYVSSLVWALVVAVIAPILFYSG
TGVRRNKTITCYDTTADEYLRSYFVYSMCTTVFMFCIPFIVILGCYGLIVKALIYKDLDN
SPLRRKSIYLVIIVLTVFAVSYLPFHVMKTLNLRARLDFQTPQMCAFNDKVYATYQVTRG
LASLNSCVDPILYFLAGDTFRRRLSRATRKSSRRSEPNVQSKSEEMTLNILTEYKQNGDT
SL
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| BDBM50102301 |
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| n/a |
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| Name | BDBM50102301 |
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| Synonyms: | 4-[4-Formyl-5-hydroxy-6-methyl-3-(2-phosphono-ethyl)-pyridin-2-ylazo]-benzoic acid | CHEMBL117766 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H16N3O7P |
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| Mol. Mass. | 393.2879 |
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| SMILES | Cc1nc(N=Nc2ccc(cc2)C(O)=O)c(CCP(O)(O)=O)c(C=O)c1O |w:5.5| |
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| Structure | 
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