| Reaction Details |
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 | Report a problem with these data |
| Target | Endoplasmin |
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| Ligand | BDBM14487 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2035398 (CHEMBL4689556) |
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| Kd | >50000±n/a nM |
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| Citation |  Tosh, DK; Brackett, CM; Jung, YH; Gao, ZG; Banerjee, M; Blagg, BSJ; Jacobson, KA Biological Evaluation of 5'-( ACS Med Chem Lett12:373-379 (2021) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Endoplasmin |
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| Name: | Endoplasmin |
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| Synonyms: | 94 kDa glucose-regulated protein | ENPL_HUMAN | GRP-94 | GRP94 | Glucose regulated protein 94kDa (Grp94) | HSP90B1 | Heat shock protein 90 kDa beta member 1 | TRA1 | Tumor rejection antigen 1 | gp96 homolog |
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| Type: | Protein |
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| Mol. Mass.: | 92417.36 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P14625 |
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| Residue: | 803 |
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| Sequence: | MRALWVLGLCCVLLTFGSVRADDEVDVDGTVEEDLGKSREGSRTDDEVVQREEEAIQLDG
LNASQIRELREKSEKFAFQAEVNRMMKLIINSLYKNKEIFLRELISNASDALDKIRLISL
TDENALSGNEELTVKIKCDKEKNLLHVTDTGVGMTREELVKNLGTIAKSGTSEFLNKMTE
AQEDGQSTSELIGQFGVGFYSAFLVADKVIVTSKHNNDTQHIWESDSNEFSVIADPRGNT
LGRGTTITLVLKEEASDYLELDTIKNLVKKYSQFINFPIYVWSSKTETVEEPMEEEEAAK
EEKEESDDEAAVEEEEEEKKPKTKKVEKTVWDWELMNDIKPIWQRPSKEVEEDEYKAFYK
SFSKESDDPMAYIHFTAEGEVTFKSILFVPTSAPRGLFDEYGSKKSDYIKLYVRRVFITD
DFHDMMPKYLNFVKGVVDSDDLPLNVSRETLQQHKLLKVIRKKLVRKTLDMIKKIADDKY
NDTFWKEFGTNIKLGVIEDHSNRTRLAKLLRFQSSHHPTDITSLDQYVERMKEKQDKIYF
MAGSSRKEAESSPFVERLLKKGYEVIYLTEPVDEYCIQALPEFDGKRFQNVAKEGVKFDE
SEKTKESREAVEKEFEPLLNWMKDKALKDKIEKAVVSQRLTESPCALVASQYGWSGNMER
IMKAQAYQTGKDISTNYYASQKKTFEINPRHPLIRDMLRRIKEDEDDKTVLDLAVVLFET
ATLRSGYLLPDTKAYGDRIERMLRLSLNIDPDAKVEEEPEEEPEETAEDTTEDTEQDEDE
EMDVGTDEEEETAKESTAEKDEL
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| BDBM14487 |
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| n/a |
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| Name | BDBM14487 |
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| Synonyms: | (2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxymethyl)oxolane-3,4-diol | Adenine-beta-D-arabinofuranoside | Adenosine | CHEMBL477 | N6-Methylado | [U-14C]adenosine | cid_191 | cid_60961 |
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| Type | Nucleoside or nucleotide |
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| Emp. Form. | C10H13N5O4 |
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| Mol. Mass. | 267.2413 |
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| SMILES | Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CO)[C@@H](O)[C@H]1O |
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| Structure | 
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