| Reaction Details |
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 | Report a problem with these data |
| Target | Protein kinase C delta type |
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| Ligand | BDBM50554605 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2050085 (CHEMBL4704784) |
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| Ki | 0.740000±n/a nM |
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| Citation |  Kobayashi, T; Yanagita, RC; Irie, K Synthesis and biological activities of simplified aplysiatoxin analogs focused on the CH/? interaction. Bioorg Med Chem Lett30:0 (2020) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Protein kinase C delta type |
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| Name: | Protein kinase C delta type |
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| Synonyms: | KPCD_MOUSE | Pkcd | Prkcd | Protein kinase C delta | Protein kinase C delta type | nPKC-delta |
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| Type: | PROTEIN |
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| Mol. Mass.: | 77554.99 |
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| Organism: | Mus musculus |
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| Description: | ChEMBL_1351519 |
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| Residue: | 674 |
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| Sequence: | MAPFLRISFNSYELGSLQVEDEASQPFCAVKMKEALSTERGKTLVQKKPTMYPEWKTTFD
AHIYEGRVIQIVLMRAAEDPVSEVTVGVSVLAERCKKNNGKAEFWLDLQPQAKVLMCVQY
FLEDGDCKQSMRSEEEAKFPTMNRRGAIKQAKIHYIKNHEFIATFFGQPTFCSVCKEFVW
GLNKQGYKCRQCNAAIHKKCIDKIIGRCTGTATNSRDTIFQKERFNIDMPHRFKVYNYMS
PTFCDHCGSLLWGLVKQGLKCEDCGMNVHHKCREKVANLCGINQKLLAEALNQVTQRSSR
KLDTTESVGIYQGFEKKPEVSGSDILDNNGTYGKIWEGSTRCTLENFTFQKVLGKGSFGK
VLLAELKGKDKYFAIKCLKKDVVLIDDDVECTMVEKRVLALAWESPFLTHLICTFQTKDH
LFFVMEFLNGGDLMFHIQDKGRFELYRATFYAAEIICGLQFLHSKGIIYRDLKLDNVMLD
RDGHIKIADFGMCKENIFGEGRASTFCGTPDYIAPEILQGLKYSFSVDWWSFGVLLYEML
IGQSPFHGDDEDELFESIRVDTPHYPRWITKESKDIMEKLFERDPDKRLGVTGNIRIHPF
FKTINWSLLEKRKVEPPFKPKVKSPSDYSNFDPEFLNEKPQLSFSDKNLIDSMDQEAFHG
FSFVNPKFEQFLDI
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| BDBM50554605 |
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| n/a |
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| Name | BDBM50554605 |
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| Synonyms: | CHEMBL4755092 |
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| Type | Small organic molecule |
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| Emp. Form. | C39H48O8 |
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| Mol. Mass. | 644.7936 |
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| SMILES | [H][C@@]12CCC(C)(C)[C@]3(C[C@]([H])(OC(=O)C[C@H](CO)OC(=O)C1)[C@H](C)[C@@H](CCCCc1cccc4cc(OCc5ccccc5)ccc14)O3)O2 |r| |
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| Structure | 
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