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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Retinoic acid receptor RXR-gamma | ||
| Ligand | BDBM50092055 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | ChEBML_70528 | ||
| Ki | >6000±n/a nM | ||
| Citation |  Walker, JR; Alshafie, G; Abou-Issa, H; Curley, RW An improved synthesis of the C-linked glucuronide of N-(4-hydroxyphenyl)retinamide. Bioorg Med Chem Lett12:2447-50 (2002) [PubMed] | ||
| More Info.: | Get all data from this article, Assay Method | ||
| Retinoic acid receptor RXR-gamma | |||
| Name: | Retinoic acid receptor RXR-gamma | ||
| Synonyms: | NR2B3 | Nuclear receptor subfamily 2 group B member 3 | RXRG | RXRG_HUMAN | Retinoic acid receptor RXR-gamma | Retinoid X receptor gamma | Retinoid X receptor gamma/retinoic acid receptor alpha | ||
| Type: | PROTEIN | ||
| Mol. Mass.: | 50878.26 | ||
| Organism: | Homo sapiens (Human) | ||
| Description: | ChEMBL_197216 | ||
| Residue: | 463 | ||
| Sequence: |
| ||
| BDBM50092055 | |||
| n/a | |||
| Name | BDBM50092055 | ||
| Synonyms: | (2E,4E,6E,8E)-3,7-Dimethyl-9-(2,6,6-trimethyl-cyclohex-1-enyl)-nona-2,4,6,8-tetraenoic acid (4-hydroxy-phenyl)-amide | (2E,4E,6E,8E)-N-(4-hydroxyphenyl)-3,7-dimethyl-9-(2,6,6-trimethylcyclohex-1-enyl)nona-2,4,6,8-tetraenamide | 3,7-Dimethyl-9-(2,6,6-trimethyl-cyclohex-1-enyl)-nona-2,4,6,8-tetraenoic acid (4-hydroxy-phenyl)-amide | 4-hydroxyphenyl retinamide | CHEMBL7301 | FENRETINIDE | N-(4-HYDROXYPHENYL)ALL-TRANS RETINAMIDE | N-(4-hydroxyphenyl)-retinamide | N-(4-hydroxyphenyl)retinamide | N-(4-hydroxyphenyl)retinamide, 4-HPR | ||
| Type | Small organic molecule | ||
| Emp. Form. | C26H33NO2 | ||
| Mol. Mass. | 391.5457 | ||
| SMILES | C\C(\C=C\C1=C(C)CCCC1(C)C)=C/C=C/C(/C)=C/C(=O)Nc1ccc(O)cc1 |c:4| | ||
| Structure | 
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