| Reaction Details |
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 | Report a problem with these data |
| Target | G-protein coupled receptor 84 |
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| Ligand | BDBM50556779 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2057186 (CHEMBL4712187) |
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| IC50 | 4.8±n/a nM |
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| Citation |  Chen, LH; Zhang, Q; Xie, X; Nan, FJ Modulation of the G-Protein-Coupled Receptor 84 (GPR84) by Agonists and Antagonists. J Med Chem63:15399-15409 (2020) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| G-protein coupled receptor 84 |
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| Name: | G-protein coupled receptor 84 |
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| Synonyms: | EX33 | G-protein coupled receptor 84 | GPR84 | GPR84_HUMAN | Inflammation-related G-protein coupled receptor EX33 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 43726.73 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_116040 |
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| Residue: | 396 |
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| Sequence: | MWNSSDANFSCYHESVLGYRYVAVSWGVVVAVTGTVGNVLTLLALAIQPKLRTRFNLLIA
NLTLADLLYCTLLQPFSVDTYLHLHWRTGATFCRVFGLLLFASNSVSILTLCLIALGRYL
LIAHPKLFPQVFSAKGIVLALVSTWVVGVASFAPLWPIYILVPVVCTCSFDRIRGRPYTT
ILMGIYFVLGLSSVGIFYCLIHRQVKRAAQALDQYKLRQASIHSNHVARTDEAMPGRFQE
LDSRLASGGPSEGISSEPVSAATTQTLEGDSSEVGDQINSKRAKQMAEKSPPEASAKAQP
IKGARRAPDSSSEFGKVTRMCFAVFLCFALSYIPFLLLNILDARVQAPRVVHMLAANLTW
LNGCINPVLYAAMNRQFRQAYGSILKRGPRSFHRLH
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| BDBM50556779 |
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| n/a |
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| Name | BDBM50556779 |
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| Synonyms: | CHEMBL3715656 |
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| Type | Small organic molecule |
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| Emp. Form. | C26H25N3O4 |
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| Mol. Mass. | 443.4944 |
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| SMILES | O=c1nc(OCC2COCCO2)cc2-c3ccc(cc3CCn12)C#CCNc1ccccc1 |
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| Structure | 
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