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Target5-hydroxytryptamine receptor 1B
LigandBDBM50094968
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1805 (CHEMBL616778)
Ki>10000±n/a nM
Citation Ferretti, GDukat, MGiannella, MPiergentili, APigini, MQuaglia, WDamaj, MIMartin, BRGlennon, RA Homoazanicotine: a structure-affinity study for nicotinic acetylcholine (nACh) receptor binding. J Med Chem45:4724-31 (2002) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
5-hydroxytryptamine receptor 1B
Name:5-hydroxytryptamine receptor 1B
Synonyms:5-HT-1B | 5-HT1B | 5-hydroxytryptamine receptor 1B (5HT1B) | 5HT1B_RAT | 5ht1b | Htr1b | Serotonin 1 (5-HT1) receptor | Serotonin 1B/1D receptor | Serotonin receptor 1B
Type:Protein
Mol. Mass.:43173.33
Organism:Rattus norvegicus (Rat)
Description:P28564
Residue:386
Sequence:
MEEQGIQCAPPPPATSQTGVPLANLSHNCSADDYIYQDSIALPWKVLLVALLALITLATT
LSNAFVIATVYRTRKLHTPANYLIASLAVTDLLVSILVMPISTMYTVTGRWTLGQVVCDF
WLSSDITCCTASIMHLCVIALDRYWAITDAVDYSAKRTPKRAAIMIVLVWVFSISISLPP
FFWRQAKAEEEVLDCFVNTDHVLYTVYSTVGAFYLPTLLLIALYGRIYVEARSRILKQTP
NKTGKRLTRAQLITDSPGSTSSVTSINSRVPEVPSESGSPVYVNQVKVRVSDALLEKKKL
MAARERKATKTLGIILGAFIVCWLPFFIISLVMPICKDACWFHMAIFDFFNWLGYLNSLI
NPIIYTMSNEDFKQAFHKLIRFKCTG
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50094968
n/a
NameBDBM50094968
Synonyms:3-(1-Methyl-4,5-dihydro-1H-imidazol-2-ylmethyl)-pyridine | CHEMBL313631
TypeSmall organic molecule
Emp. Form.C10H13N3
Mol. Mass.175.2303
SMILESCN1CCN=C1Cc1cccnc1 |c:4|
Structure
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