| Reaction Details |
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 | Report a problem with these data |
| Target | Beta-galactoside alpha-2,6-sialyltransferase 1 |
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| Ligand | BDBM50559954 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2070763 (CHEMBL4726297) |
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| Ki | 8500±n/a nM |
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| Citation |  Montgomery, AP; Dobie, C; Szabo, R; Hallam, L; Ranson, M; Yu, H; Skropeta, D Design, synthesis and evaluation of carbamate-linked uridyl-based inhibitors of human ST6Gal I. Bioorg Med Chem28:0 (2020) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Beta-galactoside alpha-2,6-sialyltransferase 1 |
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| Name: | Beta-galactoside alpha-2,6-sialyltransferase 1 |
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| Synonyms: | Alpha 2,6-ST 1 | B-cell antigen CD75 | Beta-galactoside alpha-2,6-sialyltransferase 1 | CMP-N-acetylneuraminate-beta-galactosamide-alpha-2,6-sialyltransferase 1 | SIAT1 | SIAT1_HUMAN | ST6GAL1 | ST6Gal I | ST6GalI | Sialyltransferase 1 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 46622.19 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_109837 |
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| Residue: | 406 |
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| Sequence: | MIHTNLKKKFSCCVLVFLLFAVICVWKEKKKGSYYDSFKLQTKEFQVLKSLGKLAMGSDS
QSVSSSSTQDPHRGRQTLGSLRGLAKAKPEASFQVWNKDSSSKNLIPRLQKIWKNYLSMN
KYKVSYKGPGPGIKFSAEALRCHLRDHVNVSMVEVTDFPFNTSEWEGYLPKESIRTKAGP
WGRCAVVSSAGSLKSSQLGREIDDHDAVLRFNGAPTANFQQDVGTKTTIRLMNSQLVTTE
KRFLKDSLYNEGILIVWDPSVYHSDIPKWYQNPDYNFFNNYKTYRKLHPNQPFYILKPQM
PWELWDILQEISPEEIQPNPPSSGMLGIIIMMTLCDQVDIYEFLPSKRKTDVCYYYQKFF
DSACTMGAYHPLLYEKNLVKHLNQGTDEDIYLLGKATLPGFRTIHC
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| BDBM50559954 |
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| n/a |
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| Name | BDBM50559954 |
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| Synonyms: | CHEMBL4755740 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H18N3Na2O10PS |
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| Mol. Mass. | 557.379 |
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| SMILES | n/a |
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| Structure | 
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