| Reaction Details |
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 | Report a problem with these data |
| Target | Chemerin-like receptor 1 |
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| Ligand | BDBM50560519 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2072271 (CHEMBL4727805) |
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| IC50 | 130±n/a nM |
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| Citation |  Imaizumi, T; Otsubo, S; Komai, M; Takada, H; Maemoto, M; Kobayashi, A; Otsubo, N The design, synthesis and evaluation of 2-aminobenzoxazole analogues as potent and orally efficacious ChemR23 inhibitors. Bioorg Med Chem28:0 (2020) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Chemerin-like receptor 1 |
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| Name: | Chemerin-like receptor 1 |
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| Synonyms: | CHEMR23 | CHEMR23 | CMKLR1 | CML1_HUMAN | Chemokine-like receptor 1 | DEZ | G-protein coupled receptor ChemR23 | G-protein coupled receptor DEZ |
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| Type: | PROTEIN |
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| Mol. Mass.: | 42333.62 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_100822 |
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| Residue: | 373 |
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| Sequence: | MRMEDEDYNTSISYGDEYPDYLDSIVVLEDLSPLEARVTRIFLVVVYSIVCFLGILGNGL
VIIIATFKMKKTVNMVWFLNLAVADFLFNVFLPIHITYAAMDYHWVFGTAMCKISNFLLI
HNMFTSVFLLTIISSDRCISVLLPVWSQNHRSVRLAYMACMVIWVLAFFLSSPSLVFRDT
ANLHGKISCFNNFSLSTPGSSSWPTHSQMDPVGYSRHMVVTVTRFLCGFLVPVLIITACY
LTIVCKLQRNRLAKTKKPFKIIVTIIITFFLCWCPYHTLNLLELHHTAMPGSVFSLGLPL
ATALAIANSCMNPILYVFMGQDFKKFKVALFSRLVNALSEDTGHSSYPSHRSFTKMSSMN
ERTSMNERETGML
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| BDBM50560519 |
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| n/a |
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| Name | BDBM50560519 |
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| Synonyms: | CHEMBL4779379 |
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| Type | Small organic molecule |
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| Emp. Form. | C31H31N7O |
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| Mol. Mass. | 517.6241 |
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| SMILES | CCCCN([C@H](C)c1ccc(cc1)-c1ccccc1-c1nnn[nH]1)c1nc2c(cccc2o1)-c1cccn1C |r| |
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| Structure | 
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