| Reaction Details |
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 | Report a problem with these data |
| Target | Melanocortin receptor 4 |
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| Ligand | BDBM50561609 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2075512 (CHEMBL4731046) |
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| EC50 | >100000±n/a nM |
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| Citation |  Ericson, MD; Freeman, KT; Haskell-Luevano, C Peptoid NPhe ACS Med Chem Lett11:1942-1948 (2020) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Melanocortin receptor 4 |
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| Name: | Melanocortin receptor 4 |
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| Synonyms: | MC4-R | MC4R_MOUSE | Mc4r |
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| Type: | PROTEIN |
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| Mol. Mass.: | 36964.43 |
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| Organism: | Mus musculus |
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| Description: | ChEMBL_1498850 |
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| Residue: | 332 |
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| Sequence: | MNSTHHHGMYTSLHLWNRSSYGLHGNASESLGKGHPDGGCYEQLFVSPEVFVTLGVISLL
ENILVIVAIAKNKNLHSPMYFFICSLAVADMLVSVSNGSETIVITLLNSTDTDAQSFTVN
IDNVIDSVICSSLLASICSLLSIAVDRYFTIFYALQYHNIMTVRRVGIIISCIWAACTVS
GVLFIIYSDSSAVIICLISMFFTMLVLMASLYVHMFLMARLHIKRIAVLPGTGTIRQGTN
MKGAITLTILIGVFVVCWAPFFLHLLFYISCPQNPYCVCFMSHFNLYLILIMCNAVIDPL
IYALRSQELRKTFKEIICFYPLGGICELSSRY
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| BDBM50561609 |
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| n/a |
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| Name | BDBM50561609 |
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| Synonyms: | CHEMBL4753150 |
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| Type | Small organic molecule |
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| Emp. Form. | C49H64N12O8 |
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| Mol. Mass. | 949.1081 |
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| SMILES | [H][C@@]12CCCN1C(=O)[C@@]1([H])CCCN1C(=O)CN(Cc1ccccc1)C(=O)[C@H](C)NC(=O)[C@H](CN)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCCNC(N)=N)NC2=O |r| |
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| Structure | 
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