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TargetNeuropeptide FF receptor 1
LigandBDBM50565185
Substrate/Competitorn/a
Meas. Tech.ChEMBL_2090997 (CHEMBL4772260)
Ki 13±n/a nM
Citation Nguyen, TMarusich, JLi, JXZhang, Y Neuropeptide FF and Its Receptors: Therapeutic Applications and Ligand Development. J Med Chem63:12387-12402 (2020) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Neuropeptide FF receptor 1
Name:Neuropeptide FF receptor 1
Synonyms:G-protein coupled receptor 147 | GPR147 | NPFF1 | NPFF1_HUMAN | NPFFR1 | RFamide-related peptide receptor OT7T022
Type:PROTEIN
Mol. Mass.:47840.07
Organism:Homo sapiens (Human)
Description:ChEMBL_1474637
Residue:430
Sequence:
MEGEPSQPPNSSWPLSQNGTNTEATPATNLTFSSYYQHTSPVAAMFIVAYALIFLLCMVG
NTLVCFIVLKNRHMHTVTNMFILNLAVSDLLVGIFCMPTTLVDNLITGWPFDNATCKMSG
LVQGMSVSASVFTLVAIAVERFRCIVHPFREKLTLRKALVTIAVIWALALLIMCPSAVTL
TVTREEHHFMVDARNRSYPLYSCWEAWPEKGMRRVYTTVLFSHIYLAPLALIVVMYARIA
RKLCQAPGPAPGGEEAADPRASRRRARVVHMLVMVALFFTLSWLPLWALLLLIDYGQLSA
PQLHLVTVYAFPFAHWLAFFNSSANPIIYGYFNENFRRGFQAAFRARLCPRPSGSHKEAY
SERPGGLLHRRVFVVVRPSDSGLPSESGPSSGAPRPGRLPLRNGRVAHHGLPREGPGCSH
LPLTIPAWDI
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  Blast E-value cutoff:
BDBM50565185
n/a
NameBDBM50565185
Synonyms:CHEMBL4777535
TypeSmall organic molecule
Emp. Form.C11H12N4
Mol. Mass.200.2398
SMILESCc1cc(NC(N)=N)nc2ccccc12
Structure
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