| Reaction Details |
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 | Report a problem with these data |
| Target | Somatostatin receptor type 5 |
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| Ligand | BDBM50136767 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_200855 (CHEMBL807064) |
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| IC50 | >10000±n/a nM |
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| Citation |  Erchegyi, J; Waser, B; Schaer, JC; Cescato, R; Brazeau, JF; Rivier, J; Reubi, JC Novel sst(4)-selective somatostatin (SRIF) agonists. 3. Analogues amenable to radiolabeling. J Med Chem46:5597-605 (2003) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Somatostatin receptor type 5 |
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| Name: | Somatostatin receptor type 5 |
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| Synonyms: | SOMATOSTATIN SST5 | SS-5-R | SS5-R | SS5R | SSR5_HUMAN | SSTR5 | Somatostatin receptor type 5 (SSTR5) |
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| Type: | Enzyme |
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| Mol. Mass.: | 39218.02 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P35346 |
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| Residue: | 364 |
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| Sequence: | MEPLFPASTPSWNASSPGAASGGGDNRTLVGPAPSAGARAVLVPVLYLLVCAAGLGGNTL
VIYVVLRFAKMKTVTNIYILNLAVADVLYMLGLPFLATQNAASFWPFGPVLCRLVMTLDG
VNQFTSVFCLTVMSVDRYLAVVHPLSSARWRRPRVAKLASAAAWVLSLCMSLPLLVFADV
QEGGTCNASWPEPVGLWGAVFIIYTAVLGFFAPLLVICLCYLLIVVKVRAAGVRVGCVRR
RSERKVTRMVLVVVLVFAGCWLPFFTVNIVNLAVALPQEPASAGLYFFVVILSYANSCAN
PVLYGFLSDNFRQSFQKVLCLRKGSGAKDADATEPRPDRIRQQQEATPPAHRAAANGLMQ
TSKL
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| BDBM50136767 |
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| n/a |
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| Name | BDBM50136767 |
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| Synonyms: | 2-[4-(5,7-Difluoro-2-phenyl-1H-indol-3-yl)-butyrylamino]-5-guanidino-pentanoic acid methyl ester | CHEMBL153158 | L-803,087 |
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| Type | Small organic molecule |
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| Emp. Form. | C25H29F2N5O3 |
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| Mol. Mass. | 485.5263 |
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| SMILES | COC(=O)C(CCCNC(N)=N)NC(=O)CCCc1c([nH]c2c(F)cc(F)cc12)-c1ccccc1 |
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| Structure | 
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