| Reaction Details |
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 | Report a problem with these data |
| Target | Syndecan-2 |
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| Ligand | BDBM50574549 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2122626 (CHEMBL4831859) |
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| IC50 | >200000±n/a nM |
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| Citation |  Garcia, M; Hoffer, L; Leblanc, R; Benmansour, F; Feracci, M; Derviaux, C; Egea-Jimenez, AL; Roche, P; Zimmermann, P; Morelli, X; Barral, K Fragment-based drug design targeting syntenin PDZ2 domain involved in exosomal release and tumour spread. Eur J Med Chem223:0 (2021) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Syndecan-2 |
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| Name: | Syndecan-2 |
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| Synonyms: | CD_antigen=CD362 | Fibroglycan | HSPG | HSPG1 | Heparan sulfate proteoglycan core protein | SDC2 | SDC2_HUMAN | SYND2 | Syndecan-2 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 22149.57 |
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| Organism: | Homo sapiens |
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| Description: | ChEMBL_120518 |
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| Residue: | 201 |
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| Sequence: | MRRAWILLTLGLVACVSAESRAELTSDKDMYLDNSSIEEASGVYPIDDDDYASASGSGAD
EDVESPELTTSRPLPKILLTSAAPKVETTTLNIQNKIPAQTKSPEETDKEKVHLSDSERK
MDPAEEDTNVYTEKHSDSLFKRTEVLAAVIAGGVIGFLFAIFLILLLVYRMRKKDEGSYD
LGERKPSSAAYQKAPTKEFYA
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| BDBM50574549 |
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| n/a |
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| Name | BDBM50574549 |
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| Synonyms: | CHEMBL4875884 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H27NO5S |
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| Mol. Mass. | 429.529 |
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| SMILES | CC(C)[C@H](NC(=O)CCSc1ccc(cc1)-c1ccc(CCC(O)=O)cc1)C(O)=O |r| |
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| Structure | 
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