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TargetMelatonin receptor
LigandBDBM50140302
Substrate/Competitorn/a
Meas. Tech.ChEBML_105264
Ki 0.140000±n/a nM
Citation Sun LQChen JTakaki KJohnson GIben LMahle CDRyan EXu C Design and synthesis of benzoxazole derivatives as novel melatoninergic ligands. Bioorg Med Chem Lett 14:1197-200 (2004) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Melatonin receptor
Name:Melatonin receptor
Synonyms:MTNR1B | Mel-1B-R | Mel1b melatonin receptor | Melatonin 1B | Melatonin receptor | Melatonin receptor type 1B | Melatonin receptor type 2 (MT2)
Type:Enzyme
Mol. Mass.:40203.54
Organism:Homo sapiens (Human)
Description:P49286
Residue:362
Sequence:
MSENGSFANCCEAGGWAVRPGWSGAGSARPSRTPRPPWVAPALSAVLIVTTAVDVVGNLL
VILSVLRNRKLRNAGNLFLVSLALADLVVAFYPYPLILVAIFYDGWALGEEHCKASAFVM
GLSVIGSVFNITAIAINRYCYICHSMAYHRIYRRWHTPLHICLIWLLTVVALLPNFFVGS
LEYDPRIYSCTFIQTASTQYTAAVVVIHFLLPIAVVSFCYLRIWVLVLQARRKAKPESRL
CLKPSDLRSFLTMFVVFVIFAICWAPLNCIGLAVAINPQEMAPQIPEGLFVTSYLLAYFN
SCLNAIVYGLLNQNFRREYKRILLALWNPRHCIQDASKGSHAEGLQSPAPPIIGVQHQAD
AL
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  Blast E-value cutoff:
BDBM50140302
n/a
NameBDBM50140302
Synonyms:CHEMBL279343 | Cyclopropanecarboxylic acid [(1R,2R)-2-(2-propyl-2,3-dihydro-benzooxazol-7-yl)-cyclopropylmethyl]-amide
TypeSmall organic molecule
Emp. Form.C18H24N2O2
Mol. Mass.300.3954
SMILESCCCC1Nc2cccc([C@@H]3C[C@H]3CNC(=O)C3CC3)c2O1
Structure
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