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TargetMu-type opioid receptor (Mu)
LigandBDBM50143266
Substrate/Competitorn/a
Meas. Tech.ChEMBL_148096
Ki 85±n/a nM
Citation Van Cauwenberghe SSimonin FCluzeau JBecker JALubell WDTourwé D Structure-activity study of the ORL1 antagonist Ac-Arg-D-Cha-Qaa-D-Arg-D-p-ClPhe-NH2. J Med Chem 47:1864-7 (2004) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Mu-type opioid receptor (Mu)
Name:Delta opioid receptor
Synonyms:n/a
Type:n/a
Mol. Mass.:40382.98
Organism:Homo sapiens (Human)
Description:n/a
Residue:372
Sequence:
MEPAPSAGAELQPPLFANASDAYPSACPSAGANASGPPGARSASSLALAIAITALYSAVC
AVGLLGNVLVMFGIVRYTKMKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELL
CKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVG
VPIMVMAVTRPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRL
RSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDIDRRDPLVVAAL
HLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRKPCGRPDPSSFSRAREATARERVTAC
TPSDGPGGGAAA
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  Blast E-value cutoff:
BDBM50143266
n/a
NameBDBM50143266
Synonyms:7-[(R)-2-((S)-2-Acetylamino-5-ureido-pentanoylamino)-3-cyclohexyl-propionylamino]-6-oxo-octahydro-quinolizine-4-carboxylic acid {(R)-1-[1-carbamoyl-2-((R)-4-chloro-phenyl)-ethylcarbamoyl]-4-guanidino-butyl}-amide | CHEMBL3144465
TypeSmall organic molecule
Emp. Form.C40H62ClN11O7
Mol. Mass.844.443
SMILES[H][C@]12CCC[C@H](N1C(=O)[C@H](CC2)NC(=O)[C@@H](CC1CCCCC1)NC(=O)CCCCNC(N)=N)C(=O)N[C@H](CCCNC(N)=O)C(=O)N[C@H](Cc1ccc(Cl)cc1)C(N)=O
Structure
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