| Reaction Details |
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 | Report a problem with these data |
| Target | Nuclear receptor subfamily 4 group A member 2 |
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| Ligand | BDBM50577601 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2130664 (CHEMBL4840093) |
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| IC50 | 31000±n/a nM |
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| Citation |  Zaienne, D; Willems, S; Schierle, S; Heering, J; Merk, D Development and Profiling of Inverse Agonist Tools for the Neuroprotective Transcription Factor Nurr1. J Med Chem64:15126-15140 (2021) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Nuclear receptor subfamily 4 group A member 2 |
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| Name: | Nuclear receptor subfamily 4 group A member 2 |
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| Synonyms: | NOT | NR4A2 | NR4A2_HUMAN | NURR1 | TINUR |
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| Type: | PROTEIN |
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| Mol. Mass.: | 66603.77 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_453027 |
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| Residue: | 598 |
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| Sequence: | MPCVQAQYGSSPQGASPASQSYSYHSSGEYSSDFLTPEFVKFSMDLTNTEITATTSLPSF
STFMDNYSTGYDVKPPCLYQMPLSGQQSSIKVEDIQMHNYQQHSHLPPQSEEMMPHSGSV
YYKPSSPPTPTTPGFQVQHSPMWDDPGSLHNFHQNYVATTHMIEQRKTPVSRLSLFSFKQ
SPPGTPVSSCQMRFDGPLHVPMNPEPAGSHHVVDGQTFAVPNPIRKPASMGFPGLQIGHA
SQLLDTQVPSPPSRGSPSNEGLCAVCGDNAACQHYGVRTCEGCKGFFKRTVQKNAKYVCL
ANKNCPVDKRRRNRCQYCRFQKCLAVGMVKEVVRTDSLKGRRGRLPSKPKSPQEPSPPSP
PVSLISALVRAHVDSNPAMTSLDYSRFQANPDYQMSGDDTQHIQQFYDLLTGSMEIIRGW
AEKIPGFADLPKADQDLLFESAFLELFVLRLAYRSNPVEGKLIFCNGVVLHRLQCVRGFG
EWIDSIVEFSSNLQNMNIDISAFSCIAALAMVTERHGLKEPKRVEELQNKIVNCLKDHVT
FNNGGLNRPNYLSKLLGKLPELRTLCTQGLQRIFYLKLEDLVPPPAIIDKLFLDTLPF
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| BDBM50577601 |
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| n/a |
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| Name | BDBM50577601 |
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| Synonyms: | CHEMBL4850618 |
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| Type | Small organic molecule |
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| Emp. Form. | C12H13NO2 |
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| Mol. Mass. | 203.2371 |
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| SMILES | CCn1cc(C(=O)OC)c2ccccc12 |
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| Structure | 
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