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TargetGlucagon-like peptide 1 receptor
LigandBDBM50152768
Substrate/Competitorn/a
Meas. Tech.ChEMBL_304159 (CHEMBL829998)
EC50>1000±n/a nM
Citation Léger, RThibaudeau, KRobitaille, MQuraishi, Ovan Wyk, PBousquet-Gagnon, NCarette, JCastaigne, JPBridon, DP Identification of CJC-1131-albumin bioconjugate as a stable and bioactive GLP-1(7-36) analog. Bioorg Med Chem Lett14:4395-8 (2004) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Glucagon-like peptide 1 receptor
Name:Glucagon-like peptide 1 receptor
Synonyms:GLP-1 receptor | GLP-1-R | GLP-1R | GLP1R | GLP1R_HUMAN | Glucagon-like peptide 1 receptor | Glucagon-like peptide 1 receptor (GLP-1)
Type:Enzyme
Mol. Mass.:53035.78
Organism:Homo sapiens (Human)
Description:P43220
Residue:463
Sequence:
MAGAPGPLRLALLLLGMVGRAGPRPQGATVSLWETVQKWREYRRQCQRSLTEDPPPATDL
FCNRTFDEYACWPDGEPGSFVNVSCPWYLPWASSVPQGHVYRFCTAEGLWLQKDNSSLPW
RDLSECEESKRGERSSPEEQLLFLYIIYTVGYALSFSALVIASAILLGFRHLHCTRNYIH
LNLFASFILRALSVFIKDAALKWMYSTAAQQHQWDGLLSYQDSLSCRLVFLLMQYCVAAN
YYWLLVEGVYLYTLLAFSVLSEQWIFRLYVSIGWGVPLLFVVPWGIVKYLYEDEGCWTRN
SNMNYWLIIRLPILFAIGVNFLIFVRVICIVVSKLKANLMCKTDIKCRLAKSTLTLIPLL
GTHEVIFAFVMDEHARGTLRFIKLFTELSFTSFQGLMVAILYCFVNNEVQLEFRKSWERW
RLEHLHIQRDSSMKPLKCPTSSLSSGATAGSSMYTATCQASCS
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  Blast E-value cutoff:
BDBM50152768
n/a
NameBDBM50152768
Synonyms:CHEMBL265428 | GLP-17-(7-36) derivative
TypeSmall organic molecule
Emp. Form.C162H242N42O51
Mol. Mass.3593.9057
SMILESn/a
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least: