| Reaction Details |
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 | Report a problem with these data |
| Target | Adenosine receptor A3 |
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| Ligand | BDBM50585019 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2161287 (CHEMBL5046037) |
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| Ki | >10000±n/a nM |
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| Citation |  Tang, ML; Wen, ZH; Wang, JH; Wang, ML; Zhang, H; Liu, XH; Jin, L; Chang, J Discovery of Pyridone-Substituted Triazolopyrimidine Dual A ACS Med Chem Lett13:436-442 (2022) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Adenosine receptor A3 |
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| Name: | Adenosine receptor A3 |
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| Synonyms: | A3 adenosine receptor (hA3) | AA3R_HUMAN | ADORA3 | Adenosine A3 receptor (A3AR) |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 36197.32 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P0DMS8 |
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| Residue: | 318 |
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| Sequence: | MPNNSTALSLANVTYITMEIFIGLCAIVGNVLVICVVKLNPSLQTTTFYFIVSLALADIA
VGVLVMPLAIVVSLGITIHFYSCLFMTCLLLIFTHASIMSLLAIAVDRYLRVKLTVRYKR
VTTHRRIWLALGLCWLVSFLVGLTPMFGWNMKLTSEYHRNVTFLSCQFVSVMRMDYMVYF
SFLTWIFIPLVVMCAIYLDIFYIIRNKLSLNLSNSKETGAFYGREFKTAKSLFLVLFLFA
LSWLPLSIINCIIYFNGEVPQLVLYMGILLSHANSMMNPIVYAYKIKKFKETYLLILKAC
VVCHPSDSLDTSIEKNSE
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| BDBM50585019 |
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| n/a |
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| Name | BDBM50585019 |
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| Synonyms: | CHEMBL5074137 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H13N7O |
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| Mol. Mass. | 319.3207 |
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| SMILES | Cn1cc(ccc1=O)-c1cnc(N)n2nc(nc12)-c1ccccn1 |
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| Structure | 
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