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TargetLysophosphatidic acid receptor 2
LigandBDBM50170854
Substrate/Competitorn/a
Meas. Tech.ChEMBL_310431 (CHEMBL834057)
EC50 3100±n/a nM
Citation Durgam, GGVirag, TWalker, MDTsukahara, RYasuda, SLiliom, Kvan Meeteren, LAMoolenaar, WHWilke, NSiess, WTigyi, GMiller, DD Synthesis, structure-activity relationships, and biological evaluation of fatty alcohol phosphates as lysophosphatidic acid receptor ligands, activators of PPARgamma, and inhibitors of autotaxin. J Med Chem48:4919-30 (2005) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Lysophosphatidic acid receptor 2
Name:Lysophosphatidic acid receptor 2
Synonyms:EDG4 | LPA receptor 2 | LPA-2 | LPA2 | LPAR2 | LPAR2_HUMAN | Lysophosphatidic acid receptor 2 | Lysophosphatidic acid receptor Edg-4
Type:PROTEIN
Mol. Mass.:39103.44
Organism:Homo sapiens (Human)
Description:ChEMBL_1451385
Residue:351
Sequence:
MVIMGQCYYNETIGFFYNNSGKELSSHWRPKDVVVVALGLTVSVLVLLTNLLVIAAIASN
RRFHQPIYYLLGNLAAADLFAGVAYLFLMFHTGPRTARLSLEGWFLRQGLLDTSLTASVA
TLLAIAVERHRSVMAVQLHSRLPRGRVVMLIVGVWVAALGLGLLPAHSWHCLCALDRCSR
MAPLLSRSYLAVWALSSLLVFLLMVAVYTRIFFYVRRRVQRMAEHVSCHPRYRETTLSLV
KTVVIILGAFVVCWTPGQVVLLLDGLGCESCNVLAVEKYFLLLAEANSLVNAAVYSCRDA
EMRRTFRRLLCCACLRQSTRESVHYTSSAQGGASTRIMLPENGHPLMDSTL
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  Blast E-value cutoff:
BDBM50170854
n/a
NameBDBM50170854
Synonyms:CHEMBL187711 | Phosphoric acid monododecyl ester
TypeSmall organic molecule
Emp. Form.C12H27O4P
Mol. Mass.266.3141
SMILESCCCCCCCCCCCCOP(O)(O)=O
Structure
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