| Reaction Details |
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 | Report a problem with these data |
| Target | Lysophosphatidic acid receptor 2 |
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| Ligand | BDBM50170858 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_310431 (CHEMBL834057) |
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| EC50 | 717±n/a nM |
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| Citation |  Durgam, GG; Virag, T; Walker, MD; Tsukahara, R; Yasuda, S; Liliom, K; van Meeteren, LA; Moolenaar, WH; Wilke, N; Siess, W; Tigyi, G; Miller, DD Synthesis, structure-activity relationships, and biological evaluation of fatty alcohol phosphates as lysophosphatidic acid receptor ligands, activators of PPARgamma, and inhibitors of autotaxin. J Med Chem48:4919-30 (2005) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Lysophosphatidic acid receptor 2 |
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| Name: | Lysophosphatidic acid receptor 2 |
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| Synonyms: | EDG4 | LPA receptor 2 | LPA-2 | LPA2 | LPAR2 | LPAR2_HUMAN | Lysophosphatidic acid receptor 2 | Lysophosphatidic acid receptor Edg-4 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 39103.44 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1451385 |
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| Residue: | 351 |
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| Sequence: | MVIMGQCYYNETIGFFYNNSGKELSSHWRPKDVVVVALGLTVSVLVLLTNLLVIAAIASN
RRFHQPIYYLLGNLAAADLFAGVAYLFLMFHTGPRTARLSLEGWFLRQGLLDTSLTASVA
TLLAIAVERHRSVMAVQLHSRLPRGRVVMLIVGVWVAALGLGLLPAHSWHCLCALDRCSR
MAPLLSRSYLAVWALSSLLVFLLMVAVYTRIFFYVRRRVQRMAEHVSCHPRYRETTLSLV
KTVVIILGAFVVCWTPGQVVLLLDGLGCESCNVLAVEKYFLLLAEANSLVNAAVYSCRDA
EMRRTFRRLLCCACLRQSTRESVHYTSSAQGGASTRIMLPENGHPLMDSTL
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| BDBM50170858 |
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| n/a |
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| Name | BDBM50170858 |
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| Synonyms: | CHEMBL190349 | Phosphoric acid mono-((E)-dodec-9-enyl) ester |
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| Type | Small organic molecule |
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| Emp. Form. | C12H25O4P |
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| Mol. Mass. | 264.2983 |
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| SMILES | CC\C=C\CCCCCCCCOP(O)(O)=O |
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| Structure | 
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