| Reaction Details |
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 | Report a problem with these data |
| Target | Adenosine receptor A3 |
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| Ligand | BDBM50597191 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2223068 (CHEMBL5136402) |
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| Kd | 55±n/a nM |
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| Citation |  Suchankova, A; Stampelou, M; Koutsouki, K; Pousias, A; Dhingra, L; Barkan, K; Pouli, N; Marakos, P; Tenta, R; Kolocouris, A; Lougiakis, N; Ladds, G Discovery of a High Affinity Adenosine A ACS Med Chem Lett13:923-934 (2022) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Adenosine receptor A3 |
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| Name: | Adenosine receptor A3 |
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| Synonyms: | A3 adenosine receptor (hA3) | AA3R_HUMAN | ADORA3 | Adenosine A3 receptor (A3AR) |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 36197.32 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P0DMS8 |
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| Residue: | 318 |
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| Sequence: | MPNNSTALSLANVTYITMEIFIGLCAIVGNVLVICVVKLNPSLQTTTFYFIVSLALADIA
VGVLVMPLAIVVSLGITIHFYSCLFMTCLLLIFTHASIMSLLAIAVDRYLRVKLTVRYKR
VTTHRRIWLALGLCWLVSFLVGLTPMFGWNMKLTSEYHRNVTFLSCQFVSVMRMDYMVYF
SFLTWIFIPLVVMCAIYLDIFYIIRNKLSLNLSNSKETGAFYGREFKTAKSLFLVLFLFA
LSWLPLSIINCIIYFNGEVPQLVLYMGILLSHANSMMNPIVYAYKIKKFKETYLLILKAC
VVCHPSDSLDTSIEKNSE
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| BDBM50597191 |
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| n/a |
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| Name | BDBM50597191 |
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| Synonyms: | CHEMBL5195631 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H17N5 |
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| Mol. Mass. | 315.3718 |
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| SMILES | Cn1nc(-c2ccccc2)c2cnnc(NCc3ccccc3)c12 |
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| Structure | 
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