Reaction Details |
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Target | Trace amine-associated receptor 1 |
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Ligand | BDBM50181793 |
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Substrate/Competitor | n/a |
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Meas. Tech. | ChEMBL_332032 (CHEMBL859597) |
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EC50 | 333±n/a nM |
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Citation | Hart, ME; Suchland, KL; Miyakawa, M; Bunzow, JR; Grandy, DK; Scanlan, TS Trace amine-associated receptor agonists: synthesis and evaluation of thyronamines and related analogues. J Med Chem49:1101-12 (2006) [PubMed] Article |
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More Info.: | Get all data from this article, Assay Method |
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Trace amine-associated receptor 1 |
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Name: | Trace amine-associated receptor 1 |
Synonyms: | TAAR1_RAT | Ta1 | Taar1 | Tar1 | Trace amine receptor 1 (TARR1) | Trace amine-associated receptor 1 | Trace amine-associated receptor 1 (TAAR1) | Trace amine-associated receptor1 | Trar1 |
Type: | Enzyme |
Mol. Mass.: | 38034.73 |
Organism: | Rattus norvegicus (Rat) |
Description: | Q923Y9 |
Residue: | 332 |
Sequence: | MHLCHNSANISHTNSNWSRDVRASLYSLISLIILTTLVGNLIVIISISHFKQLHTPTNWL
LHSMAVVDFLLGCLVMPYSMVRTVEHCWYFGELFCKLHTSTDIMLSSASILHLAFISIDR
YYAVCDPLRYKAKINLAAIFVMILISWSLPAVFAFGMIFLELNLEGVEELYHNQVFCLRG
CFPFFSKVSGVLAFMTSFYIPGSVMLFVYYRIYFIAKGQARSINRANLQVGLEGESRAPQ
SKETKAAKTLGIMVGVFLLCWCPFFFCMVLDPFLGYVIPPTLNDTLNWFGYLNSAFNPMV
YAFFYPWFRRALKMVLFGKIFQKDSSRSKLFL
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BDBM50181793 |
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n/a |
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Name | BDBM50181793 |
Synonyms: | CHEMBL202548 | O-(m,m-dimethoxy)benzyl-tyramine |
Type | Small organic molecule |
Emp. Form. | C17H21NO3 |
Mol. Mass. | 287.3535 |
SMILES | COc1cc(COc2ccc(CCN)cc2)cc(OC)c1 |
Structure |
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