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TargetTrace amine-associated receptor 1
LigandBDBM50181807
Substrate/Competitorn/a
Meas. Tech.ChEMBL_332033 (CHEMBL859598)
EC50>1000±n/a nM
Citation Hart, MESuchland, KLMiyakawa, MBunzow, JRGrandy, DKScanlan, TS Trace amine-associated receptor agonists: synthesis and evaluation of thyronamines and related analogues. J Med Chem49:1101-12 (2006) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Trace amine-associated receptor 1
Name:Trace amine-associated receptor 1
Synonyms:TAAR1_MOUSE | Ta1 | Taar1 | Tar1 | Trace amine receptor 1 (TARR1) | Trace amine-associated receptor 1 (TAAR1) | Trace amine-associated receptor1 | Trar1
Type:Protein
Mol. Mass.:37635.41
Organism:Mus musculus (Mouse)
Description:Q923Y8
Residue:332
Sequence:
MHLCHAITNISHRNSDWSREVQASLYSLMSLIILATLVGNLIVIISISHFKQLHTPTNWL
LHSMAIVDFLLGCLIMPCSMVRTVERCWYFGEILCKVHTSTDIMLSSASIFHLAFISIDR
YCAVCDPLRYKAKINISTILVMILVSWSLPAVYAFGMIFLELNLKGVEELYRSQVSDLGG
CSPFFSKVSGVLAFMTSFYIPGSVMLFVYYRIYFIAKGQARSINRTNVQVGLEGKSQAPQ
SKETKAAKTLGIMVGVFLVCWCPFFLCTVLDPFLGYVIPPSLNDALYWFGYLNSALNPMV
YAFFYPWFRRALKMVLLGKIFQKDSSRSKLFL
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  Blast E-value cutoff:
BDBM50181807
n/a
NameBDBM50181807
Synonyms:CHEMBL202172 | O-(2',3',4',5',6'-pentafluoro)benzyl-tyramine
TypeSmall organic molecule
Emp. Form.C15H12F5NO
Mol. Mass.317.2539
SMILESNCCc1ccc(OCc2c(F)c(F)c(F)c(F)c2F)cc1
Structure
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