| Reaction Details |
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 | Report a problem with these data |
| Target | Trace amine-associated receptor 1 |
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| Ligand | BDBM50181794 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_332032 (CHEMBL859597) |
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| EC50 | >1000±n/a nM |
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| Citation |  Hart, ME; Suchland, KL; Miyakawa, M; Bunzow, JR; Grandy, DK; Scanlan, TS Trace amine-associated receptor agonists: synthesis and evaluation of thyronamines and related analogues. J Med Chem49:1101-12 (2006) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Trace amine-associated receptor 1 |
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| Name: | Trace amine-associated receptor 1 |
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| Synonyms: | TAAR1_RAT | Ta1 | Taar1 | Tar1 | Trace amine receptor 1 (TARR1) | Trace amine-associated receptor 1 | Trace amine-associated receptor 1 (TAAR1) | Trace amine-associated receptor1 | Trar1 |
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| Type: | Enzyme |
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| Mol. Mass.: | 38034.73 |
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| Organism: | Rattus norvegicus (Rat) |
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| Description: | Q923Y9 |
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| Residue: | 332 |
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| Sequence: | MHLCHNSANISHTNSNWSRDVRASLYSLISLIILTTLVGNLIVIISISHFKQLHTPTNWL
LHSMAVVDFLLGCLVMPYSMVRTVEHCWYFGELFCKLHTSTDIMLSSASILHLAFISIDR
YYAVCDPLRYKAKINLAAIFVMILISWSLPAVFAFGMIFLELNLEGVEELYHNQVFCLRG
CFPFFSKVSGVLAFMTSFYIPGSVMLFVYYRIYFIAKGQARSINRANLQVGLEGESRAPQ
SKETKAAKTLGIMVGVFLLCWCPFFFCMVLDPFLGYVIPPTLNDTLNWFGYLNSAFNPMV
YAFFYPWFRRALKMVLFGKIFQKDSSRSKLFL
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| BDBM50181794 |
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| n/a |
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| Name | BDBM50181794 |
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| Synonyms: | CHEMBL425223 | O-(p-trifluoromethyl)benzyl-3-iodotyramine |
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| Type | Small organic molecule |
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| Emp. Form. | C16H15F3INO |
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| Mol. Mass. | 421.1961 |
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| SMILES | NCCc1ccc(OCc2ccc(cc2)C(F)(F)F)c(I)c1 |
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| Structure | 
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