Reaction Details |
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Target | Trace amine-associated receptor 1 |
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Ligand | BDBM50181805 |
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Substrate/Competitor | n/a |
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Meas. Tech. | ChEMBL_332033 (CHEMBL859598) |
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EC50 | >1000±n/a nM |
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Citation | Hart, ME; Suchland, KL; Miyakawa, M; Bunzow, JR; Grandy, DK; Scanlan, TS Trace amine-associated receptor agonists: synthesis and evaluation of thyronamines and related analogues. J Med Chem49:1101-12 (2006) [PubMed] Article |
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More Info.: | Get all data from this article, Assay Method |
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Trace amine-associated receptor 1 |
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Name: | Trace amine-associated receptor 1 |
Synonyms: | TAAR1_MOUSE | Ta1 | Taar1 | Tar1 | Trace amine receptor 1 (TARR1) | Trace amine-associated receptor 1 (TAAR1) | Trace amine-associated receptor1 | Trar1 |
Type: | Protein |
Mol. Mass.: | 37635.41 |
Organism: | Mus musculus (Mouse) |
Description: | Q923Y8 |
Residue: | 332 |
Sequence: | MHLCHAITNISHRNSDWSREVQASLYSLMSLIILATLVGNLIVIISISHFKQLHTPTNWL
LHSMAIVDFLLGCLIMPCSMVRTVERCWYFGEILCKVHTSTDIMLSSASIFHLAFISIDR
YCAVCDPLRYKAKINISTILVMILVSWSLPAVYAFGMIFLELNLKGVEELYRSQVSDLGG
CSPFFSKVSGVLAFMTSFYIPGSVMLFVYYRIYFIAKGQARSINRTNVQVGLEGKSQAPQ
SKETKAAKTLGIMVGVFLVCWCPFFLCTVLDPFLGYVIPPSLNDALYWFGYLNSALNPMV
YAFFYPWFRRALKMVLLGKIFQKDSSRSKLFL
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BDBM50181805 |
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n/a |
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Name | BDBM50181805 |
Synonyms: | 3',5'-diiodothyronamine | CHEMBL201001 |
Type | Small organic molecule |
Emp. Form. | C14H13I2NO2 |
Mol. Mass. | 481.0675 |
SMILES | NCCc1ccc(Oc2cc(I)c(O)c(I)c2)cc1 |
Structure |
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