| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Trace amine-associated receptor 1 |
|---|
| Ligand | BDBM50181812 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_332033 (CHEMBL859598) |
|---|
| EC50 | 32.5±n/a nM |
|---|
| Citation |  Hart, ME; Suchland, KL; Miyakawa, M; Bunzow, JR; Grandy, DK; Scanlan, TS Trace amine-associated receptor agonists: synthesis and evaluation of thyronamines and related analogues. J Med Chem49:1101-12 (2006) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Trace amine-associated receptor 1 |
|---|
| Name: | Trace amine-associated receptor 1 |
|---|
| Synonyms: | TAAR1_MOUSE | Ta1 | Taar1 | Tar1 | Trace amine receptor 1 (TARR1) | Trace amine-associated receptor 1 (TAAR1) | Trace amine-associated receptor1 | Trar1 |
|---|
| Type: | Protein |
|---|
| Mol. Mass.: | 37635.41 |
|---|
| Organism: | Mus musculus (Mouse) |
|---|
| Description: | Q923Y8 |
|---|
| Residue: | 332 |
|---|
| Sequence: | MHLCHAITNISHRNSDWSREVQASLYSLMSLIILATLVGNLIVIISISHFKQLHTPTNWL
LHSMAIVDFLLGCLIMPCSMVRTVERCWYFGEILCKVHTSTDIMLSSASIFHLAFISIDR
YCAVCDPLRYKAKINISTILVMILVSWSLPAVYAFGMIFLELNLKGVEELYRSQVSDLGG
CSPFFSKVSGVLAFMTSFYIPGSVMLFVYYRIYFIAKGQARSINRTNVQVGLEGKSQAPQ
SKETKAAKTLGIMVGVFLVCWCPFFLCTVLDPFLGYVIPPSLNDALYWFGYLNSALNPMV
YAFFYPWFRRALKMVLLGKIFQKDSSRSKLFL
|
|
|
|---|
| BDBM50181812 |
|---|
| n/a |
|---|
| Name | BDBM50181812 |
|---|
| Synonyms: | CHEMBL382580 | O-(p-fluoro)phenyl-3-iodotyramine |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C15H15FINO |
|---|
| Mol. Mass. | 371.1886 |
|---|
| SMILES | CNCCc1ccc(Oc2ccc(F)cc2)c(I)c1 |
|---|
| Structure | 
|
|---|
Search and Browse
