Ki Summary

Reaction Details

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Target

Solute carrier family 15 member 2

Ligand

BDBM50190616

Substrate/Competitor

n/a

Meas. Tech.

ChEMBL_370529 (CHEMBL871420)

3700±n/a nM

Citation

Biegel, A; Gebauer, S; Brandsch, M; Neubert, K; Thondorf, I Structural requirements for the substrates of the H+/peptide cotransporter PEPT2 determined by three-dimensional quantitative structure-activity relationship analysis. J Med Chem49:4286-96 (2006) [PubMed] Article

More Info.:

Get all data from this article, Assay Method

Solute carrier family 15 member 2

Name:

Solute carrier family 15 member 2

Synonyms:

Oligopeptide transporter, kidney isoform | Pept2 | S15A2_RAT | Slc15a2

Type:

PROTEIN

Mol. Mass.:

81331.63

Organism:

Rattus norvegicus

Description:

ChEMBL_838253

Residue:

729

Sequence:

MNPFQKNESKETLFSPVSTEEMLPRPPSPPKKSPPKIFGSSYPVSIAFIVVNEFCERFSY
YGMKAVLTLYFLYFLHWNEDTSTSVYHAFSSLCYFTPILGAAIADSWLGKFKTIIYLSLV
YVLGHVFKSLGAIPILGGKMLHTILSLVGLSLIALGTGGIKPCVAAFGGDQFEEEHAEAR
TRYFSVFYLAINAGSLISTFITPMLRGDVKCFGQDCYALAFGVPGLLMVLALVVFAMGSK
MYRKPPPEGNIVAQVIKCIWFALCNRFRNRSGDLPKRQHWLDWAAEKYPKHLIADVKALT
RVLFLYIPLPMFWALLDQQGSRWTLQANKMNGDLGFFVLQPDQMQVLNPFLVLIFIPLFD
LVIYRLISKCRINFSSLRKMAVGMILACLAFAVAALVETKINGMIHPQPASQEIFLQVLN
LADGDVKVTVLGSRNNSLLVESVSSFQNTTHYSKLHLEAKSQDLHFHLKYNSLSVHNDHS
VEEKNCYQLLIHQDGESISSMLVKDTGIKPANGMAAIRFINTLHKDLNISLDTDAPLSVG
KDYGVSAYRTVLRGKYPAVHCETEDKVFSLDLGQLDFGTTYLFVITNITSQGLQAWKAED
IPVNKLSIAWQLPQYVLVTAAEVMFSVTGLEFSYSQAPSSMKSVLQAAWLLTVAVGNIIV
LVVAQFSGLAQWAEFVLFSCLLLVVCLIFSVMAYYYVPLKSEDTREATDKQIPAVQGNMI
NLETKNTRL

BDBM50190616

n/a

Name

BDBM50190616

Synonyms:

(S)-2-((S)-2-benzamido-3-phenylpropanamido)propanoic acid | CHEMBL214174

Type

Small organic molecule

Emp. Form.

C19H20N2O4

Mol. Mass.

340.3731

SMILES

C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccccc1)C(O)=O

Structure