| Reaction Details |
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 | Report a problem with these data |
| Target | P2Y purinoceptor 6 |
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| Ligand | BDBM50405421 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2265211 |
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| IC50 | 1790±n/a nM |
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| Citation |  Jung, YH; Shah, Q; Lewicki, SA; Pramanik, A; Gopinatth, V; Pelletier, J; Sévigny, J; Iqbal, J; Jacobson, KA Synthesis and pharmacological characterization of multiply substituted 2H-chromene derivatives as P2Y Bioorg Med Chem Lett75:0 (2022) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| P2Y purinoceptor 6 |
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| Name: | P2Y purinoceptor 6 |
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| Synonyms: | P2RY6 | P2RY6_HUMAN | P2Y purinoceptor 6 | P2Y6 | Pyrimidinergic receptor P2Y6 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 36452.29 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1511151 |
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| Residue: | 328 |
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| Sequence: | MEWDNGTGQALGLPPTTCVYRENFKQLLLPPVYSAVLAAGLPLNICVITQICTSRRALTR
TAVYTLNLALADLLYACSLPLLIYNYAQGDHWPFGDFACRLVRFLFYANLHGSILFLTCI
SFQRYLGICHPLAPWHKRGGRRAAWLVCVAVWLAVTTQCLPTAIFAATGIQRNRTVCYDL
SPPALATHYMPYGMALTVIGFLLPFAALLACYCLLACRLCRQDGPAEPVAQERRGKAARM
AVVVAAAFAISFLPFHITKTAYLAVRSTPGVPCTVLEAFAAAYKGTRPFASANSVLDPIL
FYFTQKKFRRRPHELLQKLTAKWQRQGR
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| BDBM50405421 |
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| n/a |
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| Name | BDBM50405421 |
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| Synonyms: | CHEMBL5279730 |
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| Type | Small organic molecule |
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| Emp. Form. | C10H5ClF3NO3 |
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| Mol. Mass. | 279.6 |
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| SMILES | [O-][N+](=O)C1=Cc2cc(Cl)ccc2OC1C(F)(F)F |t:3| |
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| Structure | 
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