| Reaction Details |
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 | Report a problem with these data |
| Target | D(2) dopamine receptor |
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| Ligand | BDBM85067 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2275348 |
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| Ki | 199±n/a nM |
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| Citation |  Giorgioni, G; Del Bello, F; Pavleti?, P; Quaglia, W; Botticelli, L; Cifani, C; Micioni Di Bonaventura, E; Micioni Di Bonaventura, MV; Piergentili, A Recent findings leading to the discovery of selective dopamine D Eur J Med Chem212:0 (2021) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| D(2) dopamine receptor |
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| Name: | D(2) dopamine receptor |
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| Synonyms: | D(2) dopamine receptor | DOPAMINE D2 | DOPAMINE D2 Long | DOPAMINE D2 Short | DRD2 | DRD2_HUMAN | Dopamine D2 receptor | Dopamine D2 receptor (D2) | Dopamine D2 receptor (D2R) | Dopamine D2A | Dopamine2-like | d2 |
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| Type: | Cell-surface receptors |
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| Mol. Mass.: | 50647.10 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P14416 |
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| Residue: | 443 |
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| Sequence: | MDPLNLSWYDDDLERQNWSRPFNGSDGKADRPHYNYYATLLTLLIAVIVFGNVLVCMAVS
REKALQTTTNYLIVSLAVADLLVATLVMPWVVYLEVVGEWKFSRIHCDIFVTLDVMMCTA
SILNLCAISIDRYTAVAMPMLYNTRYSSKRRVTVMISIVWVLSFTISCPLLFGLNNADQN
ECIIANPAFVVYSSIVSFYVPFIVTLLVYIKIYIVLRRRRKRVNTKRSSRAFRAHLRAPL
KGNCTHPEDMKLCTVIMKSNGSFPVNRRRVEAARRAQELEMEMLSSTSPPERTRYSPIPP
SHHQLTLPDPSHHGLHSTPDSPAKPEKNGHAKDHPKIAKIFEIQTMPNGKTRTSLKTMSR
RKLSQQKEKKATQMLAIVLGVFIICWLPFFITHILNIHCDCNIPPVLYSAFTWLGYVNSA
VNPIIYTTFNIEFRKAFLKILHC
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| BDBM85067 |
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| n/a |
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| Name | BDBM85067 |
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| Synonyms: | CAS_170856-41-4 | CHEMBL81330 | PNU 96415E | PNU-96415E |
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| Type | Small organic molecule |
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| Emp. Form. | C21H25FN2O |
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| Mol. Mass. | 340.4344 |
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| SMILES | Fc1ccc(cc1)N1CCN(CCC2OCCc3ccccc23)CC1 |
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| Structure | 
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