| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Dipeptidyl peptidase 9 |
|---|
| Ligand | BDBM50118931 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_492002 (CHEMBL938685) |
|---|
| IC50 | >1000000±n/a nM |
|---|
| Citation |  Van der Veken, P; De Meester, I; Dubois, V; Soroka, A; Van Goethem, S; Maes, MB; Brandt, I; Lambeir, AM; Chen, X; Haemers, A; Scharpé, S; Augustyns, K Inhibitors of dipeptidyl peptidase 8 and dipeptidyl peptidase 9. Part 1: identification of dipeptide derived leads. Bioorg Med Chem Lett18:4154-8 (2008) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Dipeptidyl peptidase 9 |
|---|
| Name: | Dipeptidyl peptidase 9 |
|---|
| Synonyms: | DPP9 | DPP9_HUMAN | DPRP-2 | DPRP2 | Dipeptidyl peptidase 9 (DDP9) | Dipeptidyl peptidase 9 (DPP-9) | Dipeptidyl peptidase 9 (DPP9) | Dipeptidyl peptidase IV-related protein 2 | Dipeptidyl peptidase IX | Dipeptidyl peptidase IX (DDP-IX) | Dipeptidyl peptidase-like protein 9 |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 98260.70 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | Q86TI2 |
|---|
| Residue: | 863 |
|---|
| Sequence: | MATTGTPTADRGDAAATDDPAARFQVQKHSWDGLRSIIHGSRKYSGLIVNKAPHDFQFVQ
KTDESGPHSHRLYYLGMPYGSRENSLLYSEIPKKVRKEALLLLSWKQMLDHFQATPHHGV
YSREEELLRERKRLGVFGITSYDFHSESGLFLFQASNSLFHCRDGGKNGFMVSPMKPLEI
KTQCSGPRMDPKICPADPAFFSFINNSDLWVANIETGEERRLTFCHQGLSNVLDDPKSAG
VATFVIQEEFDRFTGYWWCPTASWEGSEGLKTLRILYEEVDESEVEVIHVPSPALEERKT
DSYRYPRTGSKNPKIALKLAEFQTDSQGKIVSTQEKELVQPFSSLFPKVEYIARAGWTRD
GKYAWAMFLDRPQQWLQLVLLPPALFIPSTENEEQRLASARAVPRNVQPYVVYEEVTNVW
INVHDIFYPFPQSEGEDELCFLRANECKTGFCHLYKVTAVLKSQGYDWSEPFSPGEDEFK
CPIKEEIALTSGEWEVLARHGSKIWVNEETKLVYFQGTKDTPLEHHLYVVSYEAAGEIVR
LTTPGFSHSCSMSQNFDMFVSHYSSVSTPPCVHVYKLSGPDDDPLHKQPRFWASMMEAAS
CPPDYVPPEIFHFHTRSDVRLYGMIYKPHALQPGKKHPTVLFVYGGPQVQLVNNSFKGIK
YLRLNTLASLGYAVVVIDGRGSCQRGLRFEGALKNQMGQVEIEDQVEGLQFVAEKYGFID
LSRVAIHGWSYGGFLSLMGLIHKPQVFKVAIAGAPVTVWMAYDTGYTERYMDVPENNQHG
YEAGSVALHVEKLPNEPNRLLILHGFLDENVHFFHTNFLVSQLIRAGKPYQLQIYPNERH
SIRCPESGEHYEVTLLHFLQEYL
|
|
|
|---|
| BDBM50118931 |
|---|
| n/a |
|---|
| Name | BDBM50118931 |
|---|
| Synonyms: | 2-Amino-1-pyrrolidin-1-yl-ethanone | 2-amino-1-(pyrrolidin-1-yl)ethanone | CHEMBL97025 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C6H12N2O |
|---|
| Mol. Mass. | 128.1723 |
|---|
| SMILES | NCC(=O)N1CCCC1 |
|---|
| Structure | 
|
|---|
Search and Browse
