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TargetTranscriptional activator protein TraR
LigandBDBM50265900
Substrate/Competitorn/a
Meas. Tech.ChEMBL_543882 (CHEMBL1016857)
IC50 1600±n/a nM
Citation Geske, GDMattmann, MEBlackwell, HE Evaluation of a focused library of N-aryl L-homoserine lactones reveals a new set of potent quorum sensing modulators. Bioorg Med Chem Lett18:5978-81 (2008) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Transcriptional activator protein TraR
Name:Transcriptional activator protein TraR
Synonyms:TRAR_RHIRD | traR
Type:PROTEIN
Mol. Mass.:26741.83
Organism:Rhizobium radiobacter
Description:ChEMBL_765233
Residue:234
Sequence:
MQHWLDKLTDLAAIEGDECILKTGLADIADHFGFTGYAYLHIQHRHITAVTNYHRQWQST
YFDKKFEALDPVVKRARSRKHIFTWSGEHERPTLSKDERAFYDHASDFGIRSGITIPIKT
ANGFMSMFTMASDKPVIDLDREIDAVAAAATIGQIHARISFLRTTPTAEDAAWLDPKEAT
YLRWIAVGKTMEEIADVEGVKYNSVRVKLREAMKRFDVRSKAHLTALAIRRKLI
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50265900
n/a
NameBDBM50265900
Synonyms:(S)-3-(4-nitrophenyl)-N-(2-oxotetrahydrofuran-3-yl)propanamide | CHEMBL503238
TypeSmall organic molecule
Emp. Form.C13H14N2O5
Mol. Mass.278.2607
SMILES[O-][N+](=O)c1ccc(CCC(=O)N[C@H]2CCOC2=O)cc1 |r|
Structure
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