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TargetBaculoviral IAP repeat-containing protein 8
LigandBDBM50273698
Substrate/Competitorn/a
Meas. Tech.ChEMBL_537310
Ki 1.9±n/a nM
Citation Peng YSun HNikolovska-Coleska ZQiu SYang CYLu JCai QYi HKang SYang DWang S Potent, orally bioavailable diazabicyclic small-molecule mimetics of second mitochondria-derived activator of caspases. J Med Chem 51:8158-62 (2008) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Baculoviral IAP repeat-containing protein 8
Name:Baculoviral IAP repeat-containing protein 8
Synonyms:n/a
Type:PROTEIN
Mol. Mass.:27091.98
Organism:Homo sapiens (Human)
Description:ChEMBL_537310
Residue:236
Sequence:
MTGYEARLITFGTWMYSVNKEQLARAGFYAIGQEDKVQCFHCGGGLANWKPKEDPWEQHA
KWYPGCKYLLEEKGHEYINNIHLTRSLEGALVQTTKKTPSLTKRISDTIFPNPMLQEAIR
MGFDFKDVKKIMEERIQTSGSNYKTLEVLVADLVSAQKDTTENELNQTSLQREISPEEPL
RRLQEEKLCKICMDRHIAVVFIPCGHLVTCKQCAEAVDRCPMCSAVIDFKQRVFMS
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  Blast E-value cutoff:
BDBM50273698
n/a
NameBDBM50273698
Synonyms:(5S,8S,10aR)-3-Acetyl-N-benzhydryl-5-((S)-2-(methylamino)-propanamido)-6-oxodeca-hydro pyrrolo[1,2-a][1,5]diazocine-8-carbox-amide | CHEMBL456400
TypeSmall organic molecule
Emp. Form.C29H37N5O4
Mol. Mass.519.6352
SMILESCN[C@@H](C)C(=O)N[C@H]1CN(CC[C@H]2CC[C@H](N2C1=O)C(=O)NC(c1ccccc1)c1ccccc1)C(C)=O |r|
Structure
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