| Reaction Details |
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 | Report a problem with these data |
| Target | Thromboxane A2 receptor |
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| Ligand | BDBM50279863 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_207649 |
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| Kd | 7.5±n/a nM |
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| Citation |  Ladouceur, G; Mais, DE; Jakubowski, JA; Utterback, BG; Robertson, DW Structural homologies among thromboxane (TXA2) receptor antagonists: Minimal pharmacophoric requirements for high affinity interaction with TXA2 receptors Bioorg Med Chem Lett1:173-178 (1991) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Thromboxane A2 receptor |
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| Name: | Thromboxane A2 receptor |
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| Synonyms: | Prostanoid TP receptor | TA2R_HUMAN | TBXA2R | TXA2-R | Thromboxane | Thromboxane A2 receptor | Thromboxane Beta |
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| Type: | Enyzme |
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| Mol. Mass.: | 37445.28 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P21731 |
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| Residue: | 343 |
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| Sequence: | MWPNGSSLGPCFRPTNITLEERRLIASPWFAASFCVVGLASNLLALSVLAGARQGGSHTR
SSFLTFLCGLVLTDFLGLLVTGTIVVSQHAALFEWHAVDPGCRLCRFMGVVMIFFGLSPL
LLGAAMASERYLGITRPFSRPAVASQRRAWATVGLVWAAALALGLLPLLGVGRYTVQYPG
SWCFLTLGAESGDVAFGLLFSMLGGLSVGLSFLLNTVSVATLCHVYHGQEAAQQRPRDSE
VEMMAQLLGIMVVASVCWLPLLVFIAQTVLRNPPAMSPAGQLSRTTEKELLIYLRVATWN
QILDPWVYILFRRAVLRRLQPRLSTRPRSLSLQPQLTQRSGLQ
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| BDBM50279863 |
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| n/a |
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| Name | BDBM50279863 |
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| Synonyms: | (Z)-7-((1R,2S)-2-Benzenesulfonylamino-cyclopentyl)-hept-5-enoic acid | CHEMBL300681 |
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| Type | Small organic molecule |
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| Emp. Form. | C18H25NO4S |
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| Mol. Mass. | 351.46 |
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| SMILES | OC(=O)CCC\C=C/C[C@H]1CCC[C@@H]1NS(=O)(=O)c1ccccc1 |
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| Structure | 
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