| Reaction Details |
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 | Report a problem with these data |
| Target | Muscarinic acetylcholine receptor M1 |
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| Ligand | BDBM50280565 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_138273 |
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| EC50 | 100000±n/a nM |
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| Citation |  Tecle, H; Mirzadegan, T; Moos, WH; Moreland, DW; Pavia, MR; Schwarz, RD; Davis, RE A rationale for the design and synthesis of m1 selective muscarinic agonists. Bioorg Med Chem Lett2:821-826 (1992) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Muscarinic acetylcholine receptor M1 |
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| Name: | Muscarinic acetylcholine receptor M1 |
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| Synonyms: | ACM1_HUMAN | CHRM1 | Cholinergic receptor, muscarinic 1 | Cholinergic, muscarinic M1 |
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| Type: | Protein |
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| Mol. Mass.: | 51442.54 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P11229 |
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| Residue: | 460 |
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| Sequence: | MNTSAPPAVSPNITVLAPGKGPWQVAFIGITTGLLSLATVTGNLLVLISFKVNTELKTVN
NYFLLSLACADLIIGTFSMNLYTTYLLMGHWALGTLACDLWLALDYVASNASVMNLLLIS
FDRYFSVTRPLSYRAKRTPRRAALMIGLAWLVSFVLWAPAILFWQYLVGERTVLAGQCYI
QFLSQPIITFGTAMAAFYLPVTVMCTLYWRIYRETENRARELAALQGSETPGKGGGSSSS
SERSQPGAEGSPETPPGRCCRCCRAPRLLQAYSWKEEEEEDEGSMESLTSSEGEEPGSEV
VIKMPMVDPEAQAPTKQPPRSSPNTVKRPTKKGRDRAGKGQKPRGKEQLAKRKTFSLVKE
KKAARTLSAILLAFILTWTPYNIMVLVSTFCKDCVPETLWELGYWLCYVNSTINPMCYAL
CNKAFRDTFRLLLLCRWDKRRWRKIPKRPGSVHRTPSRQC
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| BDBM50280565 |
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| n/a |
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| Name | BDBM50280565 |
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| Synonyms: | 5-(1-Aza-bicyclo[2.2.1]hept-3-yl)-[1,2,4]oxadiazol-3-ylamine | CHEMBL314737 |
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| Type | Small organic molecule |
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| Emp. Form. | C8H12N4O |
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| Mol. Mass. | 180.2071 |
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| SMILES | Nc1noc(n1)C1CN2CCC1C2 |THB:4:6:12:10.9| |
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| Structure | 
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