| Reaction Details |
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 | Report a problem with these data |
| Target | Coagulation factor X |
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| Ligand | BDBM50280654 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_69536 |
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| IC50 | 2200±n/a nM |
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| Citation |  Sall, DJ; Berry, DR; Coffman, WJ; Craft, TJ; Denney, ML; Gifford-Moore, DS; Kellam, ML; Smith, GF Characterization of LY806303 as a potent and selective inhibitor of thrombin Bioorg Med Chem Lett2:1025-1028 (1992) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Coagulation factor X |
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| Name: | Coagulation factor X |
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| Synonyms: | Coagulation factor X | F10 | FA10_BOVIN | Factor Xa (fXa) |
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| Type: | PROTEIN |
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| Mol. Mass.: | 54498.45 |
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| Organism: | Bos taurus |
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| Description: | ChEMBL_1364435 |
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| Residue: | 492 |
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| Sequence: | MAGLLHLVLLSTALGGLLRPAGSVFLPRDQAHRVLQRARRANSFLEEVKQGNLERECLEE
ACSLEEAREVFEDAEQTDEFWSKYKDGDQCEGHPCLNQGHCKDGIGDYTCTCAEGFEGKN
CEFSTREICSLDNGGCDQFCREERSEVRCSCAHGYVLGDDSKSCVSTERFPCGKFTQGRS
RRWAIHTSEDALDASELEHYDPADLSPTESSLDLLGLNRTEPSAGEDGSQVVRIVGGRDC
AEGECPWQALLVNEENEGFCGGTILNEFYVLTAAHCLHQAKRFTVRVGDRNTEQEEGNEM
AHEVEMTVKHSRFVKETYDFDIAVLRLKTPIRFRRNVAPACLPEKDWAEATLMTQKTGIV
SGFGRTHEKGRLSSTLKMLEVPYVDRSTCKLSSSFTITPNMFCAGYDTQPEDACQGDSGG
PHVTRFKDTYFVTGIVSWGEGCARKGKFGVYTKVSNFLKWIDKIMKARAGAAGSRGHSEA
PATWTVPPPLPL
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| BDBM50280654 |
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| n/a |
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| Name | BDBM50280654 |
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| Synonyms: | (S)-5-Guanidino-2-{[(S)-1-((S)-2-methylamino-2-phenyl-acetyl)-pyrrolidine-2-carbonyl]-amino}-pentanoic acid | CHEMBL8108 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H30N6O4 |
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| Mol. Mass. | 418.49 |
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| SMILES | CN[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCNC(N)=N)C(O)=O)c1ccccc1 |
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| Structure | 
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