| Reaction Details |
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 | Report a problem with these data |
| Target | Glucagon receptor |
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| Ligand | BDBM50280717 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_219265 |
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| IC50 | 4000±n/a nM |
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| Citation |  Collins, JL; Dambek, PJ; Goldstein, SW; Faraci, W CP-99,711: a non-peptide glucagon receptor antagonist Bioorg Med Chem Lett2:915-918 (1992) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Glucagon receptor |
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| Name: | Glucagon receptor |
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| Synonyms: | GL-R | GLR_RAT | Gcgr |
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| Type: | PROTEIN |
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| Mol. Mass.: | 55053.40 |
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| Organism: | Rattus norvegicus |
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| Description: | ChEMBL_1450588 |
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| Residue: | 485 |
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| Sequence: | MLLTQLHCPYLLLLLVVLSCLPKAPSAQVMDFLFEKWKLYSDQCHHNLSLLPPPTELVCN
RTFDKYSCWPDTPPNTTANISCPWYLPWYHKVQHRLVFKRCGPDGQWVRGPRGQSWRDAS
QCQMDDDEIEVQKGVAKMYSSYQVMYTVGYSLSLGALLLALVILLGLRKLHCTRNYIHGN
LFASFVLKAGSVLVIDWLLKTRYSQKIGDDLSVSVWLSDGAVAGCRVATVIMQYGIIANY
CWLLVEGVYLYSLLSITTFSEKSFFSLYLCIGWGSPLLFVIPWVVVKCLFENVQCWTSND
NMGFWWILRIPVLLAILINFFIFVRIIHLLVAKLRAHQMHYADYKFRLARSTLTLIPLLG
VHEVVFAFVTDEHAQGTLRSTKLFFDLFFSSFQGLLVAVLYCFLNKEVQAELLRRWRRWQ
EGKALQEERMASSHGSHMAPAGTCHGDPCEKLQLMSAGSSSGTGCEPSAKTSLASSLPRL
ADSPT
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| BDBM50280717 |
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| n/a |
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| Name | BDBM50280717 |
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| Synonyms: | CHEMBL557974 | CP-99711 | N-[6,7-Dichloro-3-((E)-styryl)-quinoxalin-2-yl]-N,N',N'-trimethyl-propane-1,3-diamine; hydrochloride |
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| Type | Small organic molecule |
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| Emp. Form. | C22H24Cl2N4 |
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| Mol. Mass. | 415.359 |
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| SMILES | CN(C)CCCN(C)c1nc2cc(Cl)c(Cl)cc2nc1\C=C\c1ccccc1 |
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| Structure | 
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