Reaction Details |
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Target | Mu-type opioid receptor |
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Ligand | BDBM50281661 |
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Substrate/Competitor | n/a |
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Meas. Tech. | ChEBML_139005 |
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Ki | >10000±n/a nM |
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Citation | Higginbottom, M; Nolan, W; O'Toole, J; Ratcliffe, GS; Rees, DC; Roberts, E The design and synthesis of kappa opioid ligands based on a binding model for kappa agonists Bioorg Med Chem Lett3:841-846 (1993) Article |
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More Info.: | Get all data from this article, Assay Method |
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Mu-type opioid receptor |
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Name: | Mu-type opioid receptor |
Synonyms: | M-OR-1 | MOP | MOR-1 | MOR1 | MUOR1 | Mu Opioid Receptor | Mu opiate receptor | OPIATE Mu | OPRM1 | OPRM_HUMAN | hMOP | mu-type opioid receptor isoform MOR-1 |
Type: | G Protein-Coupled Receptor (GPCR) |
Mol. Mass.: | 44789.51 |
Organism: | Homo sapiens (Human) |
Description: | P35372 |
Residue: | 400 |
Sequence: | MDSSAAPTNASNCTDALAYSSCSPAPSPGSWVNLSHLDGNLSDPCGPNRTDLGGRDSLCP
PTGSPSMITAITIMALYSIVCVVGLFGNFLVMYVIVRYTKMKTATNIYIFNLALADALAT
STLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDF
RTPRNAKIINVCNWILSSAIGLPVMFMATTKYRQGSIDCTLTFSHPTWYWENLLKICVFI
FAFIMPVLIITVCYGLMILRLKSVRMLSGSKEKDRNLRRITRMVLVVVAVFIVCWTPIHI
YVIIKALVTIPETTFQTVSWHFCIALGYTNSCLNPVLYAFLDENFKRCFREFCIPTSSNI
EQQNSTRIRQNTRDHPSTANTVDRTNHQLENLEAETAPLP
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BDBM50281661 |
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n/a |
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Name | BDBM50281661 |
Synonyms: | 2-Oxa-7,10-diaza-bicyclo[11.3.1]heptadeca-1(17),13,15-trien-11-one | CHEMBL353264 | PD-146884 |
Type | Small organic molecule |
Emp. Form. | C14H20N2O2 |
Mol. Mass. | 248.3208 |
SMILES | O=C1Cc2cccc(OCCCCNCCN1)c2 |
Structure |
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