| Reaction Details |
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 | Report a problem with these data |
| Target | Type-1 angiotensin II receptor |
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| Ligand | BDBM50282347 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_36772 |
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| IC50 | 2200±n/a nM |
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| Citation |  Miyake, K; Matsukura, M; Yoneda, N; Hiroshima, O; Mori, N; Ishihara, H; Musha, T; Matsuoka, T; Shoji, T; Minami, N; Hamano, S; Saito, I Discovery and development of aryl-fused imidazole-based angiotensin II antagonists Bioorg Med Chem Lett4:213-218 (1994) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Type-1 angiotensin II receptor |
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| Name: | Type-1 angiotensin II receptor |
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| Synonyms: | AGTR1 | AGTR1_BOVIN | Angiotensin II type 1a (AT-1a) receptor |
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| Type: | PROTEIN |
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| Mol. Mass.: | 41107.81 |
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| Organism: | Bos taurus |
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| Description: | ChEMBL_36779 |
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| Residue: | 359 |
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| Sequence: | MILNSSTEDGIKRIQDDCPKAGRHNYIFIMIPTLYSIIFVVGIFGNSLVVIVIYFYMKLK
TVASVFLLNLALADLCFLLTLPLWAVYTAMEYRWPFGNYLCKIASASVSFNLYASVFLLT
CLSIDRYLAIVHPMKSRLRRTMLVAKVTCIIIWLLAGLASLPTIIHRNVFFIENTNITVC
AFHYESQNSTLPVGLGLTKNILGFLFPFLIILTSYTLIWKTLKKAYEIQKNKPRKDDIFK
IILAIVLFFFFSWVPHQIFTFMDVLIQLGLIRDCKIEDIVDTAMPITICLAYFNNCLNPL
FYGFLGKKFKKYFLQLLKYIPPKAKSHSNLSTKMSTLSYRPSENGNSSTKKPAPCIEVE
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| BDBM50282347 |
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| n/a |
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| Name | BDBM50282347 |
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| Synonyms: | 4-(2-Butyl-benzoimidazol-1-ylmethyl)-2-methyl-6-nitro-phenol | CHEMBL65955 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H21N3O3 |
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| Mol. Mass. | 339.3883 |
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| SMILES | CCCCc1nc2ccccc2n1Cc1cc(C)c(O)c(c1)[N+]([O-])=O |
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| Structure | 
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