| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50286105 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_136091 |
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| IC50 | 0.360000±n/a nM |
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| Citation |  Husbands, SM; Lewis, JW Morphinan cyclic imines and pyrrolidines containing a constrained phenyl group: High affinity opioid agonists Bioorg Med Chem Lett5:2969-2974 (1995) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 11165.58 |
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| Organism: | GUINEA PIG |
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| Description: | P97266 |
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| Residue: | 98 |
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| Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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| BDBM50286105 |
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| n/a |
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| Name | BDBM50286105 |
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| Synonyms: | CHEMBL318636 | Morphinan Cyclic Imine analogue |
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| Type | Small organic molecule |
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| Emp. Form. | C29H34N2O2 |
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| Mol. Mass. | 442.5925 |
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| SMILES | CO[C@]12C=C[C@]34C[C@@]1(C)[C@@H](N(C)[C@H]2C31CCN(C)C4Cc2ccc(O)cc12)c1ccccc1 |c:3,TLB:25:26:5:16.14.15,8:7:13.12:3.4,9:7:13.12:3.4,11:10:2:13.5.6,17:16:5:26.20.19,THB:4:5:26.20.19:16.14.15| |
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| Structure | 
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