| Reaction Details |
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 | Report a problem with these data |
| Target | Cannabinoid receptor 2 |
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| Ligand | BDBM50302304 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_596703 (CHEMBL1049673) |
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| EC50 | 2.8±n/a nM |
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| Citation |  Chu, GH; Saeui, CT; Worm, K; Weaver, DG; Goodman, AJ; Broadrup, RL; Cassel, JA; DeHaven, RN; LaBuda, CJ; Koblish, M; Brogdon, B; Smith, S; Le Bourdonnec, B; Dolle, RE Novel pyridine derivatives as potent and selective CB2 cannabinoid receptor agonists. Bioorg Med Chem Lett19:5931-5 (2009) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cannabinoid receptor 2 |
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| Name: | Cannabinoid receptor 2 |
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| Synonyms: | CANNABINOID CB2 | CB-2 | CB2 | CNR2_RAT | Cannabinoid CB2 receptor | Cannabinoid receptor | Cnr2 | rCB2 |
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| Type: | Enzyme |
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| Mol. Mass.: | 39366.68 |
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| Organism: | Rattus norvegicus (Rat) |
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| Description: | Q9QZN9 |
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| Residue: | 360 |
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| Sequence: | MAGCRELELTNGSNGGLEFNPMKEYMILSDAQQIAVAVLCTLMGLLSALENVAVLYLILS
SQRLRRKPSYLFIGSLAGADFLASVIFACNFVIFHVFHGVDSRNIFLLKIGSVTMTFTAS
VGSLLLTAVDRYLCLCYPPTYKALVTRGRALVALGVMWVLSALISYLPLMGWTCCPSPCS
ELFPLIPNDYLLGWLLFIAILFSGIIYTYGYVLWKAHQHVASLAEHQDRQVPGIARMRLD
VRLAKTLGLVMAVLLICWFPALALMGHSLVTTLSDKVKEAFAFCSMLCLVNSMINPIIYA
LRSGEIRSAAQHCLTGWKKYLQGLGSEGKEEAPKSSVTETEAEVKTTTGPGSRTPGCSNC
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| BDBM50302304 |
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| n/a |
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| Name | BDBM50302304 |
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| Synonyms: | 1,2-dimethyl-N-(5-methyl-4-(morpholinomethyl)pyridin-2-yl)cyclohexanecarboxamide | CHEMBL568564 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H31N3O2 |
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| Mol. Mass. | 345.479 |
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| SMILES | CC1CCCCC1(C)C(=O)Nc1cc(CN2CCOCC2)c(C)cn1 |
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| Structure | 
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