| Reaction Details |
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 | Report a problem with these data |
| Target | Cytochrome P450 2J2 |
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| Ligand | BDBM50305628 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_604540 (CHEMBL1074710) |
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| IC50 | 1400±n/a nM |
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| Citation |  Eldrup, AB; Soleymanzadeh, F; Farrow, NA; Kukulka, A; De Lombaert, S Optimization of piperidyl-ureas as inhibitors of soluble epoxide hydrolase. Bioorg Med Chem Lett20:571-5 (2010) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cytochrome P450 2J2 |
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| Name: | Cytochrome P450 2J2 |
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| Synonyms: | CP2J2_HUMAN | CYP2J2 |
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| Type: | Enzyme |
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| Mol. Mass.: | 57623.04 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P51589 |
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| Residue: | 502 |
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| Sequence: | MLAAMGSLAAALWAVVHPRTLLLGTVAFLLAADFLKRRRPKNYPPGPWRLPFLGNFFLVD
FEQSHLEVQLFVKKYGNLFSLELGDISAVLITGLPLIKEALIHMDQNFGNRPVTPMREHI
FKKNGLIMSSGQAWKEQRRFTLTALRNFGLGKKSLEERIQEEAQHLTEAIKEENGQPFDP
HFKINNAVSNIICSITFGERFEYQDSWFQQLLKLLDEVTYLEASKTCQLYNVFPWIMKFL
PGPHQTLFSNWKKLKLFVSHMIDKHRKDWNPAETRDFIDAYLKEMSKHTGNPTSSFHEEN
LICSTLDLFFAGTETTSTTLRWALLYMALYPEIQEKVQAEIDRVIGQGQQPSTAARESMP
YTNAVIHEVQRMGNIIPLNVPREVTVDTTLAGYHLPKGTMILTNLTALHRDPTEWATPDT
FNPDHFLENGQFKKREAFMPFSIGKRACLGEQLARTELFIFFTSLMQKFTFRPPNNEKLS
LKFRMGITISPVSHRLCAVPQV
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| BDBM50305628 |
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| n/a |
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| Name | BDBM50305628 |
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| Synonyms: | CHEMBL589135 | N-(2,4-dichlorobenzyl)-4-phenoxypiperidine-1-carboxamide |
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| Type | Small organic molecule |
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| Emp. Form. | C19H20Cl2N2O2 |
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| Mol. Mass. | 379.28 |
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| SMILES | Clc1ccc(CNC(=O)N2CCC(CC2)Oc2ccccc2)c(Cl)c1 |
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| Structure | 
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