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Target5-hydroxytryptamine receptor 1A (5-HT1A)
LigandBDBM50317424
Substrate/Competitorn/a
Meas. Tech.ChEMBL_631800
Ki 13050±n/a nM
Citation Nievergelt AHuonker PSchoop RAltmann KHGertsch J Identification of serotonin 5-HT1A receptor partial agonists in ginger. Bioorg Med Chem 18:3345-51 (2010) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
5-hydroxytryptamine receptor 1A (5-HT1A)
Name:5-hydroxytryptamine receptor 1A (5-HT1A)
Synonyms:5-HT-1A | 5-HT1A | 5-hydroxytryptamine receptor 1A | 5-hydroxytryptamine receptor 1A (5-HT-1A) | ADRB2RL1 | ADRBRL1 | Dopamine D2 receptor and serotonin 1a receptor | G-21 | HTR1A | Serotonin receptor 1A
Type:n/a
Mol. Mass.:46122.49
Organism:Homo sapiens (Human)
Description:n/a
Residue:422
Sequence:
MDVLSPGQGNNTTSPPAPFETGGNTTGISDVTVSYQVITSLLLGTLIFCAVLGNACVVAA
IALERSLQNVANYLIGSLAVTDLMVSVLVLPMAALYQVLNKWTLGQVTCDLFIALDVLCC
TSSILHLCAIALDRYWAITDPIDYVNKRTPRRAAALISLTWLIGFLISIPPMLGWRTPED
RSDPDACTISKDHGYTIYSTFGAFYIPLLLMLVLYGRIFRAARFRIRKTVKKVEKTGADT
RHGASPAPQPKKSVNGESGSRNWRLGVESKAGGALCANGAVRQGDDGAALEVIEVHRVGN
SKEHLPLPSEAGPTPCAPASFERKNERNAEAKRKMALARERKTVKTLGIIMGTFILCWLP
FFIVALVLPFCESSCHMPTLLGAIINWLGYSNSLLNPVIYAYFNKDFQNAFKKIIKCKFC
RQ
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  Blast E-value cutoff:
BDBM50317424
n/a
NameBDBM50317424
Synonyms:(E)-1-(4-Hydroxy-3-methoxy-phenyl)-dodec-4-en-3-one | 8-Shogaol | CHEMBL25893
TypeSmall organic molecule
Emp. Form.C19H28O3
Mol. Mass.304.4238
SMILESCCCCCCCC=CC(=O)CCc1ccc(O)c(OC)c1 |w:8.8|
Structure
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