Reaction Details |
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Target | Sigma non-opioid intracellular receptor 1 |
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Ligand | BDBM50321092 |
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Substrate/Competitor | n/a |
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Meas. Tech. | ChEMBL_637393 (CHEMBL1166326) |
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Ki | 665.3±n/a nM |
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Citation | Hajipour, AR; Fontanilla, D; Chu, UB; Arbabian, M; Ruoho, AE Synthesis and characterization of N,N-dialkyl and N-alkyl-N-aralkyl fenpropimorph-derived compounds as high affinity ligands for sigma receptors. Bioorg Med Chem18:4397-404 (2010) [PubMed] Article |
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More Info.: | Get all data from this article, Assay Method |
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Sigma non-opioid intracellular receptor 1 |
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Name: | Sigma non-opioid intracellular receptor 1 |
Synonyms: | OPRS1 | SGMR1_CAVPO | SIGMAR1 | Sigma 1-type opioid receptor | Sigma non-opioid intracellular receptor 1 | Sigma-1 receptor | Sigma1-receptor | Sigma1R | Sterol isomerase-like protein |
Type: | Protein |
Mol. Mass.: | 25307.17 |
Organism: | Cavia porcellus (Guinea pig) |
Description: | Q60492 |
Residue: | 223 |
Sequence: | MQWAVGRRWLWVALFLAAVAVLTQIVWLWLGTQNFVFQREEIAQLARQYAGLDHELAFSK
LIVELRRLHPVHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSPRHSGRY
WAEISDTIISGTFHQWREGTTKSEVFYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPS
TLGFALADTVFSTQDFLTLFYTLRVYARALQLELTTYLFGQDP
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BDBM50321092 |
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n/a |
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Name | BDBM50321092 |
Synonyms: | CHEMBL1165772 | N,N-Dioctyl-3-(4-fluorophenyl)propylamine |
Type | Small organic molecule |
Emp. Form. | C25H44FN |
Mol. Mass. | 377.622 |
SMILES | CCCCCCCCN(CCCCCCCC)CCCc1ccc(F)cc1 |
Structure |
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