| Reaction Details |
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 | Report a problem with these data |
| Target | Metallo-beta-lactamase type 2 |
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| Ligand | BDBM50322604 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_641771 (CHEMBL1177094) |
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| Ki | 7000±n/a nM |
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| Citation |  Lassaux, P; Hamel, M; Gulea, M; Delbrück, H; Mercuri, PS; Horsfall, L; Dehareng, D; Kupper, M; Frère, JM; Hoffmann, K; Galleni, M; Bebrone, C Mercaptophosphonate compounds as broad-spectrum inhibitors of the metallo-beta-lactamases. J Med Chem53:4862-76 (2010) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Metallo-beta-lactamase type 2 |
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| Name: | Metallo-beta-lactamase type 2 |
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| Synonyms: | BLAB_AERHY | Beta-lactamase | cphA |
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| Type: | PROTEIN |
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| Mol. Mass.: | 28022.56 |
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| Organism: | Aeromonas hydrophila |
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| Description: | ChEMBL_641771 |
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| Residue: | 254 |
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| Sequence: | MMKGWMKCGLAGAVVLMASFWGGSVRAAGMSLTQVSGPVYVVEDNYYVQENSMVYFGAKG
VTVVGATWTPDTARELHKLIKRVSRKPVLEVINTNYHTDRAGGNAYWKSIGAKVVSTRQT
RDLMKSDWAEIVAFTRKGLPEYPDLPLVLPNVVHDGDFTLQEGKVRAFYAGPAHTPDGIF
VYFPDEQVLYGNCILKEKLGNLSFADVKAYPQTLERLKAMKLPIKTVIGGHDSPLHGPEL
IDHYEALIKAAPQS
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| BDBM50322604 |
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| n/a |
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| Name | BDBM50322604 |
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| Synonyms: | 2-mercaptophenylphosphonic acid | CHEMBL1173336 |
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| Type | Small organic molecule |
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| Emp. Form. | C6H7O3PS |
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| Mol. Mass. | 190.157 |
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| SMILES | OP(O)(=O)c1ccccc1S |
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| Structure | 
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