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TargetOrnithine decarboxylase
LigandBDBM50005719
Substrate/Competitorn/a
Meas. Tech.ChEMBL_643973 (CHEMBL1211872)
IC50 35±n/a nM
Citation Klee, NWong, PEBaragaña, BMazouni, FEPhillips, MABarrett, MPGilbert, IH Selective delivery of 2-hydroxy APA to Trypanosoma brucei using the melamine motif. Bioorg Med Chem Lett20:4364-6 (2010) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Ornithine decarboxylase
Name:Ornithine decarboxylase
Synonyms:DCOR_RAT | Odc | Odc1
Type:PROTEIN
Mol. Mass.:51037.04
Organism:Rattus norvegicus
Description:ChEMBL_1344641
Residue:461
Sequence:
MGSFTKEEFDCHILDEGFTAKDILDQKINEVSSSDDKDAFYVADLGDVLKKHLRWLKALP
RVTPFYAVKCNDSRAIVSTLAAIGTGFDCASKTEIQLVQGLGVPPERIIYANPCKQVSQI
KYAASNGVQMMTFDSEIELMKVARAHPKAKLVLRIATDDSKAVCRLSVKFGATLKTSRLL
LERAKELNIDVIGVSFHVGSGCTDPETFVQAVSDARCVFDMGTEVGFSMYLLDIGGGFPG
SEDTKLKFEEITSVINPALDKYFPSDSGVRIIAEPGRYYVASAFTLAVNIIAKKTVWKEQ
TGSDDEDESNEQTLMYYVNDGVYGSFNCILYDHAHVKALLQKRPKPDEKYYSSSIWGPTC
DGLDRIVERCSLPEMHVGDWMLFENMGAYTVAAASTFNGFQRPNIYYVMSRSMWQLMKQI
QSHGFPPEVEEQDVGTLPMSCAQESGMDRHPAACASASINV
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  Blast E-value cutoff:
BDBM50005719
n/a
NameBDBM50005719
Synonyms:(APA)O-(3-Amino-propyl)-hydroxylamine | 3-AMINOOXY-1-AMINOPROPANE | CHEMBL1209776 | CHEMBL281021
TypeSmall organic molecule
Emp. Form.C3H10N2O
Mol. Mass.90.1243
SMILESNCCCON
Structure
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