| Reaction Details |
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 | Report a problem with these data |
| Target | Phospholipid transfer protein |
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| Ligand | BDBM50325127 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_651691 (CHEMBL1228381) |
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| IC50 | 80000±n/a nM |
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| Citation |  Ling, C; Zheng, Z; Jiang, XC; Zhong, W; Li, S Synthesis of a series of novel 2,4,5-trisubstituted selenazole compounds as potential PLTP inhibitors. Bioorg Med Chem Lett20:5123-5 (2010) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Phospholipid transfer protein |
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| Name: | Phospholipid transfer protein |
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| Synonyms: | PLTP | PLTP_HUMAN |
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| Type: | PROTEIN |
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| Mol. Mass.: | 54741.32 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_651691 |
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| Residue: | 493 |
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| Sequence: | MALFGALFLALLAGAHAEFPGCKIRVTSKALELVKQEGLRFLEQELETITIPDLRGKEGH
FYYNISEVKVTELQLTSSELDFQPQQELMLQITNASLGLRFRRQLLYWFFYDGGYINASA
EGVSIRTGLELSRDPAGRMKVSNVSCQASVSRMHAAFGGTFKKVYDFLSTFITSGMRFLL
NQQICPVLYHAGTVLLNSLLDTVPVRSSVDELVGIDYSLMKDPVASTSNLDMDFRGAFFP
LTERNWSLPNRAVEPQLQEEERMVYVAFSEFFFDSAMESYFRAGALQLLLVGDKVPHDLD
MLLRATYFGSIVLLSPAVIDSPLKLELRVLAPPRCTIKPSGTTISVTASVTIALVPPDQP
EVQLSSMTMDARLSAKMALRGKALRTQLDLRRFRIYSNHSALESLALIPLQAPLKTMLQI
GVMPMLNERTWRGVQIPLPEGINFVHEVVTNHAGFLTIGADLHFAKGLREVIEKNRPADV
RASTAPTPSTAAV
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| BDBM50325127 |
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| n/a |
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| Name | BDBM50325127 |
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| Synonyms: | CHEMBL1222598 | N-(5-benzyl-4-(4-methoxyphenyl)-1,3-selenazol-2-yl)-3,4-dimethoxybenzamide |
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| Type | Small organic molecule |
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| Emp. Form. | C26H24N2O4Se |
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| Mol. Mass. | 507.44 |
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| SMILES | COc1ccc(cc1)-c1nc(NC(=O)c2ccc(OC)c(OC)c2)[se]c1Cc1ccccc1 |
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| Structure | 
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