| Reaction Details |
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 | Report a problem with these data |
| Target | Delta-type opioid receptor |
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| Ligand | BDBM50329100 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_674208 (CHEMBL1274305) |
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| Ki | 0.14±n/a nM |
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| Citation |  Nagase, H; Nemoto, T; Matsubara, A; Saito, M; Yamamoto, N; Osa, Y; Hirayama, S; Nakajima, M; Nakao, K; Mochizuki, H; Fujii, H Design and synthesis of KNT-127, ad-opioid receptor agonist effective by systemic administration. Bioorg Med Chem Lett20:6302-5 (2010) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Delta-type opioid receptor |
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| Name: | Delta-type opioid receptor |
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| Synonyms: | DOR-1 | K56 | MSL-2 | OPIATE Delta | OPRD_MOUSE | Opioid receptors; mu and delta | Oprd1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 40577.25 |
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| Organism: | MOUSE |
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| Description: | P32300 |
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| Residue: | 372 |
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| Sequence: | MELVPSARAELQSSPLVNLSDAFPSAFPSAGANASGSPGARSASSLALAIAITALYSAVC
AVGLLGNVLVMFGIVRYTKLKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELL
CKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVG
VPIMVMAVTQPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRL
RSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDINRRDPLVVAAL
HLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRTPCGRQEPGSLRRPRQATTRERVTAC
TPSDGPGGGAAA
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| BDBM50329100 |
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| n/a |
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| Name | BDBM50329100 |
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| Synonyms: | CHEMBL1270475 |
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| Type | Small organic molecule |
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| Emp. Form. | C27H28N2O2 |
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| Mol. Mass. | 412.5234 |
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| SMILES | Oc1ccc2C[C@H]3N(CC4CC4)CC[C@@]4(Cc5nc6ccccc6cc5C[C@@]34O)c2c1 |r,THB:8:7:27:4.29.5| |
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| Structure | 
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