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TargetSigma non-opioid intracellular receptor 1
LigandBDBM36184
Substrate/Competitorn/a
Meas. Tech.ChEMBL_714958 (CHEMBL1663953)
Ki>10000±n/a nM
Citation Marrazzo, AFiorito, JZappalà, LPrezzavento, ORonsisvalle, SPasquinucci, LScoto, GMBernardini, RRonsisvalle, G Antiproliferative activity of phenylbutyrate ester of haloperidol metabolite II [(±)-MRJF4] in prostate cancer cells. Eur J Med Chem46:433-8 (2010) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Sigma non-opioid intracellular receptor 1
Name:Sigma non-opioid intracellular receptor 1
Synonyms:OPRS1 | SGMR1_CAVPO | SIGMAR1 | Sigma 1-type opioid receptor | Sigma non-opioid intracellular receptor 1 | Sigma-1 receptor | Sigma1-receptor | Sigma1R | Sterol isomerase-like protein
Type:Protein
Mol. Mass.:25307.17
Organism:Cavia porcellus (Guinea pig)
Description:Q60492
Residue:223
Sequence:
MQWAVGRRWLWVALFLAAVAVLTQIVWLWLGTQNFVFQREEIAQLARQYAGLDHELAFSK
LIVELRRLHPVHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSPRHSGRY
WAEISDTIISGTFHQWREGTTKSEVFYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPS
TLGFALADTVFSTQDFLTLFYTLRVYARALQLELTTYLFGQDP
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  Blast E-value cutoff:
BDBM36184
n/a
NameBDBM36184
Synonyms:4-phenylbutanoate
TypeGuest
Emp. Form.C10H11O2
Mol. Mass.163.1937
SMILES[O-]C(=O)CCCc1ccccc1
Structure
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